SCHEMBL2415052

SCHEMBL2415052

CNC(=O)OCc1cc(Br)n(S(=O)(=O)c2cccc(OC)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 1/20 0.43
HTR6 P50406 8/20 0.41
HDAC1 Q13547 1/20 0.41
NPC1 O15118 2/20 0.40
MET P08581 1/20 0.40
RAB9A P51151 1/20 0.40
PTGER2 P43116 1/20 0.40
MTNR1B P49286 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CHRM5 P08912 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
APOBEC3A P31941 1/20 0.39
KMT2A Q03164 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2472672 0.81 NAMPT (0.43) HDAC1CYP3A4ALDH1A1KMT2A
SCHEMBL4999263 0.80 AKR1C3 (0.44) MEP1BHTR6NPC1RAB9APTGER2
SCHEMBL4424529 0.79 HTR6 (0.44) HTR6METCYP3A4ALDH1A1PKM
SCHEMBL4999257 0.79 CHRM5 (0.50) MEP1BHTR6PTGER2CHRM5ALDH1A1
SCHEMBL2407643 0.75 CHRM5 (0.42) MEP1BHTR6HDAC1METPTGER2
SCHEMBL15730048 0.75 NPC1 (0.64) HDAC1NPC1RAB9AMTNR1BALDH1A1
SCHEMBL28715560 0.74 HTR6 (0.49) MEP1BHTR6METL3MBTL1CYP3A4
SCHEMBL28702913 0.72 MET (0.46) HTR6HDAC1METL3MBTL1CYP3A4
SCHEMBL28713092 0.72 KDM4E (0.38) HTR6METALDH1A1
SCHEMBL28936708 0.72 KDM4E (0.40) HTR6METALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed