SCHEMBL4424529

SCHEMBL4424529

COc1cccc(S(=O)(=O)n2cc(CC(C)(C)C)cc2Br)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 11/20 0.44
MET P08581 1/20 0.44
CYP3A4 P08684 1/20 0.43
LMNA P02545 2/20 0.42
HTT P42858 1/20 0.42
PKM P14618 2/20 0.41
PKLR P30613 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4412573 0.83 HTR6 (0.40) HTR6LMNAPOLB
SCHEMBL2407643 0.79 CHRM5 (0.42) HTR6METPKMALDH1A1
SCHEMBL2415052 0.79 MEP1B (0.43) HTR6METCYP3A4PKMALDH1A1
SCHEMBL4999257 0.79 CHRM5 (0.50) HTR6PKMALDH1A1
SCHEMBL28715560 0.79 HTR6 (0.49) HTR6METCYP3A4LMNAPKM
SCHEMBL4424525 0.79 MET (0.44) HTR6METCYP3A4LMNAPKM
SCHEMBL4999263 0.78 AKR1C3 (0.44) HTR6CYP3A4ALDH1A1
SCHEMBL28702913 0.77 MET (0.46) HTR6METCYP3A4LMNAPKM
SCHEMBL28713092 0.71 KDM4E (0.38) HTR6METMAPK1ALDH1A1
SCHEMBL28936708 0.71 KDM4E (0.40) HTR6METMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed