SCHEMBL28702913

SCHEMBL28702913

COc1cccc(S(=O)(=O)n2cc(C=O)cc2Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.46
HTR6 P50406 8/20 0.45
CYP3A4 P08684 1/20 0.45
HDAC1 Q13547 2/20 0.43
NFE2L2 Q16236 3/20 0.41
KEAP1 Q14145 1/20 0.41
CTSG P08311 1/20 0.41
CMA1 P23946 1/20 0.41
PKM P14618 1/20 0.41
PKLR P30613 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4424525 0.86 MET (0.44) METHTR6CYP3A4HDAC1NFE2L2
SCHEMBL1156596 0.85 PKM (0.45) HTR6HDAC1PKMPKLRHDAC3
SCHEMBL1156351 0.83 MET (0.43) METHTR6CYP3A4HDAC1HDAC3
SCHEMBL28715560 0.82 HTR6 (0.49) METHTR6CYP3A4NFE2L2KEAP1
SCHEMBL1156134 0.81 PARL (0.42) HTR6CYP3A4HDAC1HDAC3HDAC2
SCHEMBL28700638 0.80 PKM (0.40) HTR6CYP3A4HDAC1PKMHDAC3
SCHEMBL29202309 0.78 HTR6 (0.37) HTR6CYP3A4LMNAMAPK1HTR2A
SCHEMBL31187441 0.77 LMNA (0.35) HTR6PKMLMNAPOLBL3MBTL1
SCHEMBL4424529 0.77 HTR6 (0.44) METHTR6CYP3A4PKMPKLR
SCHEMBL29262662 0.76 LMNA (0.50) METLMNAMAPK1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114105962-B Sulfonamide structure-containing compound, preparation method and application thereof, pharmaceutical composition and application thereof 南京烁慧医药科技有限公司 2024-11-05 CN disclosed
CN-114105962-A Compound containing sulfonamide structure, preparation method and application thereof, and pharmaceutical composition and application thereof 南京烁慧医药科技有限公司 2022-03-01 CN disclosed