SCHEMBL24167145

SCHEMBL24167145

CC(=O)c1n[nH]c(Cc2ccccc2)n1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.53
NR1H3 Q13133 2/20 0.53
KLKB1 P03952 1/20 0.52
NPC1 O15118 1/20 0.51
POLB P06746 1/20 0.51
RAB9A P51151 1/20 0.51
ALPL P05186 2/20 0.48
RIPK1 Q13546 9/20 0.47
HDAC6 Q9UBN7 1/20 0.47
SCD O00767 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19224520 0.87 NR1H2 (0.56) NR1H2NR1H3KLKB1NPC1POLB
SCHEMBL24193687 0.84 ALPL (0.48) KLKB1ALPLRIPK1HDAC6
SCHEMBL23085471 0.84 NR1H2 (0.53) NR1H2NR1H3KLKB1NPC1POLB
SCHEMBL28824358 0.83 RNASEH1 (0.56) NR1H2NR1H3KLKB1NPC1POLB
SCHEMBL30848602 0.83 NR1H2 (0.51) NR1H2NR1H3KLKB1NPC1POLB
SCHEMBL3104472 0.82 SMN1; SMN2 (0.53) NR1H2NR1H3KLKB1NPC1POLB
SCHEMBL25586405 0.80 KLKB1 (0.55) NR1H2NR1H3KLKB1RIPK1HDAC6
SCHEMBL28042800 0.80 NR1H2 (0.49) NR1H2NR1H3KLKB1NPC1POLB
SCHEMBL31272348 0.77 ADORA3 (0.58) NR1H2NR1H3KLKB1NPC1POLB
SCHEMBL553327 0.77 TSHR (0.50) NR1H2NR1H3KLKB1NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230265100-A1 RIP1K INHIBITORS RIGEL PHARMACEUTICALS, INC. 2023-08-24 US disclosed
US-11718612-B2 Inhibitors of receptor interacting protein kinase I for the treatment of disease BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-08-08 US disclosed
US-11667643-B2 RIP1K inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2023-06-06 US disclosed
US-20220009936-A1 RIP1K INHIBITORS MIDCAP FINANCIAL TRUST 2022-01-13 US disclosed
WO-2022005898-A1 RIP1K INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2022-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11718612-B2 Inhibitors of receptor interacting protein kinase I for the treatment of disease RIPK1, RIPK2, RIPK4 NR1H2 1198/4885NR1H3 1397/4885KLKB1 3311/4885
US-20230265100-A1 RIP1K INHIBITORS RIPK1, RIPK2, RIPK3 NR1H2 1673/4885NR1H3 1797/4885KLKB1 2471/4885
US-20220009936-A1 RIP1K INHIBITORS RIPK1, RIPK2, RIPK3 NR1H2 1673/4885NR1H3 1797/4885KLKB1 2471/4885
US-11667643-B2 RIP1K inhibitors RIPK1, RIPK2, RIPK3 NR1H2 1673/4885NR1H3 1797/4885KLKB1 2471/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.