SCHEMBL2428503

SCHEMBL2428503

CC(C)(C)C1C(N)CN1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.32
GABRR1 P24046 1/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17596655 0.83
SCHEMBL2538318 0.80
SCHEMBL18979169 0.79 LMNA (0.34) POLB
SCHEMBL322778 0.79 DPP4 (0.34)
SCHEMBL4523902 0.79 DPP4 (0.34)
SCHEMBL16600622 0.79 DPP4 (0.34)
SCHEMBL322779 0.79 DPP4 (0.34)
SCHEMBL21199645 0.79
SCHEMBL28305316 0.78 POLB (0.32) POLB
SCHEMBL570338 0.78 POLB (0.32) POLBATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12528818-B2 Compositions and methods for inhibition of RAS LEIDOS BIOMEDICAL RESEARCH, INC. (US) 2026-01-20 US disclosed
US-12503452-B2 Antimicrobial compounds and methods CURZA GLOBAL, LLC (US) 2025-12-23 US disclosed
US-20250270225-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS NNSA 2025-08-28 US disclosed
US-20240383886-A1 Protein Tyrosine Phosphatase Degraders and Methods of Use Thereof ABBVIE INC. 2024-11-21 US disclosed
WO-2024213042-A1 BENZO-FUSED RING COMPOUND INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2024-10-17 WO disclosed
US-20240300964-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS THERAS, INC. 2024-09-12 US disclosed
EP-4373822-A2 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS Theras Inc. (US) 2024-05-29 EP disclosed
US-20230159491-A1 Antimicrobial Compounds and Methods NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-05-25 US disclosed
CN-115872996-A Estrogen receptor degradation agent compound and preparation method and application thereof 山东绿叶制药有限公司 2023-03-31 CN disclosed
WO-2023004102-A2 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS THERAS, INC. (US) 2023-01-26 WO disclosed
US-20130217880-A1 PURINONE DERIVATIVE ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-22 US disclosed
US-8012956-B2 Tropane compounds EXELIXIS, INC. (US) 2011-09-06 US disclosed
US-20100105651-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R&D) LIMITED (GB) 2010-04-29 US disclosed
EP-2074120-B1 TROPANE COMPOUNDS EXELIXIS INC (US) 2010-03-03 EP disclosed
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
US-20090163471-A1 Tropane compounds EXELIXIS, INC. 2009-06-25 US disclosed
WO-2009071691-A2 OXINDOLE DERIVATIVES AND THE USE THEREOF AS A MEDICATION ABBOTT GMBH & CO. KG (DE) 2009-06-11 WO disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100105651-A1 ANTAGONISTS OF SNS SODIUM CHANNELS CNR1, OPRL1, CHRNA10 POLB 4845/4885GABRR1 165/4885ATM 3571/4885
US-20130217880-A1 PURINONE DERIVATIVE BTK, KIT, SYK POLB 3032/4885GABRR1 4125/4885ATM 1557/4885
US-20230159491-A1 Antimicrobial Compounds and Methods MPO, NISCH, RPN2 POLB 108/4885GABRR1 3827/4885ATM 4286/4885
US-20250270225-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS KRAS, NRAS, HRAS POLB 1776/4885GABRR1 1003/4885ATM 3171/4885
US-20240383886-A1 Protein Tyrosine Phosphatase Degraders and Methods of Use Thereof PTPN5, PTPN1, PTPN2 POLB 4296/4885GABRR1 3293/4885ATM 810/4885
US-20240300964-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS KRAS, NRAS, HRAS POLB 1776/4885GABRR1 1003/4885ATM 3171/4885
US-20090163471-A1 Tropane compounds ADRA1B, ADRA2B, ADRB2 POLB 1234/4885GABRR1 862/4885ATM 3818/4885
US-12528818-B2 Compositions and methods for inhibition of RAS KRAS, NRAS, HRAS POLB 2275/4885GABRR1 4233/4885ATM 1051/4885
US-12503452-B2 Antimicrobial compounds and methods MPO, NISCH, RPN2 POLB 108/4885GABRR1 3827/4885ATM 4286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.