SCHEMBL24316436

SCHEMBL24316436

COc1ccc(Oc2ccc(Oc3ccc4ncc(C)c(=O)n4c3)cn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
LIPE Q05469 1/20 0.36
PIK3CA P42336 1/20 0.36
MTOR P42345 1/20 0.36
COMT P21964 1/20 0.35
NPBWR1 P48145 6/20 0.35
MCHR1 Q99705 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP2C9 P11712 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24316428 0.88 ALKBH1 (0.39) KDM4ENPBWR1MCHR1NPC1RAB9A
SCHEMBL24316624 0.80 KDM4E (0.36) KDM4EPIK3CAMTORMCHR1CYP1A2
SCHEMBL29539473 0.80 KDM4E (0.36) KDM4EPIK3CAMTORMCHR1CYP1A2
SCHEMBL24316659 0.80 ALKBH1 (0.40) KDM4ENPBWR1CYP1A2CYP3A4NPC1
SCHEMBL24316432 0.78 ACACB (0.37) PIK3CAMTORMCHR1CYP1A2CYP3A4
SCHEMBL24316545 0.77 CSF1R (0.43) KDM4EPIK3CAMTORNPBWR1NPC1
SCHEMBL24316808 0.77 POLB (0.41) KDM4EPIK3CAMTORCOMTNPBWR1
SCHEMBL24316434 0.76 CSF1R (0.53) KDM4EPIK3CAMTORNPBWR1NPC1
SCHEMBL24316565 0.75 CSF1R (0.44) KDM4EPIK3CAMTORNPBWR1NPC1
SCHEMBL32688112 0.68 KDM4E (0.56) KDM4ECYP1A2SMN1; SMN2ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057895-A1 HETEROAROMATIC COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2022-03-24 WO disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed