SCHEMBL24326280

SCHEMBL24326280

Cc1cccc(C)c1-c1cc(O)nc(NSc2cccc(N3CCCN(C(=O)OC(C)(C)C)CC3C(C)C)c2)n1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 1/20 0.34
SMARCA2 P51531 1/20 0.34
SMARCA4 P51532 1/20 0.34
PBRM1 Q86U86 1/20 0.34
TRPV3 Q8NET8 2/20 0.33
USP30 Q70CQ3 7/20 0.33
PFKFB3 Q16875 1/20 0.33
GPR119 Q8TDV5 1/20 0.32
PARP1 P09874 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
NTRK1 P04629 1/20 0.31
C5AR1 P21730 1/20 0.31
ACKR3 P25106 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24326293 0.88 SMARCA2 (0.33) SMARCA2SMARCA4PBRM1TRPV3USP30
SCHEMBL24326160 0.86 NR1I2 (0.30) SMARCA2SMARCA4PBRM1
SCHEMBL24325821 0.84 GPR119 (0.41) SMARCA2SMARCA4PBRM1GPR119MEN1
SCHEMBL24326719 0.80 GPR119 (0.34) TRPV3USP30PFKFB3GPR119PARP1
SCHEMBL24326273 0.77 GPR119 (0.37) NR1H2NR1H3GPR119
SCHEMBL24325770 0.74 TRPV3 (0.35) TRPV3USP30PFKFB3PARP1C5AR1
SCHEMBL24326398 0.74 MEN1 (0.37) NR1H2NR1H3TRPV3USP30PARP1
SCHEMBL24326126 0.72 IRAK4 (0.34) TRPV3MEN1KMT2ANTRK1
SCHEMBL24326671 0.72 IRAK4 (0.36) NR1H2NR1H3MEN1KMT2ANTRK1
SCHEMBL24325812 0.71 MAP4K1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed