SCHEMBL24336239

SCHEMBL24336239

CON(C)C(=O)c1ccn(C(=O)OC(C)(C)C)n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 9/20 0.37
MLYCD O95822 1/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
NR1H2 P55055 1/20 0.32
BCHE P06276 1/20 0.32
F2 P00734 1/20 0.32
ALOX15 P16050 1/20 0.32
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
USP30 Q70CQ3 1/20 0.31
SCD O00767 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28788197 0.79 KMT2A (0.37) GPR119KMT2AMEN1HPGDBCHE
SCHEMBL7421479 0.79 GABRG2 (0.40) KMT2AMEN1HPGDBCHENPC1
SCHEMBL26621269 0.75 MLYCD (0.42) MLYCD
SCHEMBL28155365 0.75 BCHE (0.37) GPR119KMT2AMEN1HPGDNR1H2
SCHEMBL5268457 0.74 OPRM1 (0.48) MLYCDKMT2AMEN1HPGDNPC1
SCHEMBL19384688 0.74 GPR119 (0.34) GPR119MLYCDNR1H2USP30
SCHEMBL18068142 0.73 BCHE (0.36) GPR119NR1H2BCHEF2
SCHEMBL30798637 0.72 MLYCD (0.36) MLYCD
SCHEMBL2959354 0.72 BCHE (0.38) GPR119KMT2AMEN1BCHEMAPT
SCHEMBL2013279 0.72 NOS1 (0.46) GPR119KMT2AMEN1HPGDBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11945796-B2 Substituted pyridine derivatives as SARM1 inhibitors NURA BIO, INC. (US) 2024-04-02 US disclosed
CN-116438171-A Substituted pyridine derivatives as SARM1 inhibitors 努拉生物公司 2023-07-14 CN disclosed
US-20220081417-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS SARM1 INHIBITORS NURA BIO, INC. 2022-03-17 US disclosed
US-20220081417-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS SARM1 INHIBITORS NURA BIO, INC. 2022-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11945796-B2 Substituted pyridine derivatives as SARM1 inhibitors SARM1, SARNP, ADRM1 GPR119 3596/4885MLYCD 2695/4885KMT2A 1817/4885
US-20220081417-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS SARM1 INHIBITORS SARM1, SARNP, ADRM1 GPR119 3596/4885MLYCD 2695/4885KMT2A 1817/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.