SCHEMBL24399159

SCHEMBL24399159

COc1ccc(CN2CC3(CN(C(=O)OC(C)(C)C)C3)C(=O)CC2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
KDM1A O60341 1/20 0.42
OPRM1 P35372 1/20 0.42
OPRL1 P41146 1/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
MMP1 P03956 1/20 0.40
MMP13 P45452 1/20 0.40
TP53 P04637 1/20 0.40
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
BACE1 P56817 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12543528 0.91 HDAC1 (0.51) ALDH1A1L3MBTL1HDAC6HDAC1HDAC8
SCHEMBL1963123 0.90 HDAC1 (0.43) ALDH1A1L3MBTL1HDAC6HDAC1HDAC8
SCHEMBL17761442 0.80 HDAC1 (0.54) ALDH1A1L3MBTL1HDAC6HDAC1HDAC8
SCHEMBL30801697 0.79 HDAC1 (0.45) ALDH1A1L3MBTL1HDAC6HDAC1HDAC8
SCHEMBL22770534 0.78 ALDH1A1 (0.46) ALDH1A1L3MBTL1HDAC6HDAC1HDAC8
SCHEMBL2262766 0.77 CYP3A4 (0.52) ALDH1A1L3MBTL1HDAC6HDAC1KDM1A
SCHEMBL5423537 0.76 HDAC1 (0.44) ALDH1A1L3MBTL1HDAC6HDAC1HDAC8
SCHEMBL29967631 0.76 ALDH1A1 (0.55) ALDH1A1L3MBTL1HDAC6HDAC1KDM1A
SCHEMBL1963140 0.75 AADAT (0.49) ALDH1A1L3MBTL1GAACYP3A4CYP2C19
SCHEMBL8294396 0.75 MMP1 (0.47) ALDH1A1L3MBTL1HDAC6HDAC1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022094271-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. (US) 2022-05-05 WO disclosed