SCHEMBL24439479

SCHEMBL24439479

O=C(O)c1ccc(C(=O)N2CCc3c(c(=O)oc4ccccc34)C2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTHFD2 P13995 16/20 1.00
MTHFD1 P11586 5/20 0.64
DRD4 P21917 1/20 0.64
NQO1 P15559 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30825595 1.00 MTHFD2 (1.00) MTHFD2MTHFD1DRD4NQO1
SCHEMBL5370174 0.85 MTHFD2 (0.73) MTHFD2MTHFD1DRD4
SCHEMBL10811259 0.71 MTHFD2 (0.55) MTHFD2DRD4
SCHEMBL11844405 0.69 MTHFD2 (0.88) MTHFD2
SCHEMBL5507692 0.69 MTHFD2 (0.52) MTHFD2DRD4
SCHEMBL2987838 0.67 MTHFD2 (0.54) MTHFD2
SCHEMBL7562741 0.67 KDM4E (0.60)
SCHEMBL11762718 0.67 MAOA (0.60) MTHFD2
SCHEMBL19965770 0.67 SIGMAR1 (0.56) MTHFD2
SCHEMBL3079170 0.66 MAPT (0.71) MTHFD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022104010-A1 COMBINATIONS OF METHYLENE TETRAHYDROFOLATE DEHYDROGENASE 2 (MTHFD2) INHIBITORS AND FOLATE-DEPLETING AGENTS AND METHODS USING SAME RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2022-05-19 WO disclosed