SCHEMBL24469657

SCHEMBL24469657

NC(=O)c1c(Cl)cnc2c1CCO2

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
NNMT P40261 1/20 0.33
PIM2 Q9P1W9 2/20 0.32
HSD17B10 Q99714 1/20 0.32
SIRT6 Q8N6T7 1/20 0.32
PARP1 P09874 1/20 0.31
ACHE P22303 1/20 0.31
RORC P51449 2/20 0.30
KCNH2 Q12809 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24469661 0.73 ACVRL1 (0.42) TSHRNNMTHSD17B10SIRT6
SCHEMBL21225333 0.71 TSHR (0.41) TSHRHSD17B10PARP1RORCALDH1A1
SCHEMBL29520278 0.71 TSHR (0.41) TSHRHSD17B10PARP1RORCALDH1A1
SCHEMBL28763414 0.68 POLB (0.38) HSD17B10PARP1KDM4EALDH1A1HPGD
SCHEMBL24469604 0.68 PARP1 (0.42) NNMTPARP1KDM4EL3MBTL1
SCHEMBL17371696 0.68 ALDH1A1 (0.36) ALDH1A1
SCHEMBL6282473 0.66 NNMT (0.51) TSHRNNMTPARP1LMNA
SCHEMBL30427718 0.66 NNMT (0.51) TSHRNNMTPARP1LMNA
SCHEMBL7425664 0.64 SIRT6 (0.38) TSHRNNMTHSD17B10SIRT6ALDH1A1
SCHEMBL1703067 0.63 ICAM1 (0.47) TSHRNNMTHSD17B10SIRT6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4251149-A1 MODIFIED ISOINDOLINONES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS Merck Sharp & Dohme LLC (US) 2023-10-04 EP disclosed
WO-2022115301-A1 MODIFIED ISOINDOLINONES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2022-06-02 WO disclosed
WO-2022115301-A1 MODIFIED ISOINDOLINONES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2022-06-02 WO disclosed