SCHEMBL24543294

SCHEMBL24543294

COC(=O)C1OCCc2c(Cl)ccc(F)c21

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.37
HPGD P15428 2/20 0.34
ALDH1A1 P00352 2/20 0.34
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24543296 0.86 KDM4E (0.39) ALDH1A1MAPT
SCHEMBL24542962 0.76 SIRT1 (0.38) MAPT
SCHEMBL24542958 0.76 TAS1R3 (0.36) SLC6A3ALDH1A1SLC6A4
SCHEMBL29673091 0.76 SIRT1 (0.38) MAPT
SCHEMBL24543429 0.75 ALDH1A1 (0.39) SLC6A3HPGDALDH1A1RAB9A
SCHEMBL15321005 0.67 RAB9A (0.41) SLC6A3ALDH1A1RAB9A
SCHEMBL296739 0.66 RAB9A (0.40) SLC6A3ALDH1A1RAB9A
SCHEMBL22491754 0.66 RAB9A (0.40) SLC6A3ALDH1A1RAB9A
SCHEMBL3112694 0.66 ALDH1A1 (0.35) ALDH1A1
SCHEMBL2730679 0.64 TSHR (0.34) SLC6A3HPGDALDH1A1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127827-A1 KRASG12C PROTEIN MUTATION INHIBITOR AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 上海维申医药有限公司 2022-06-23 WO disclosed