SCHEMBL24628702

SCHEMBL24628702

O=CN1CCc2cc(O)cc(C#Cc3ccccc3)c2C1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 13/20 0.39
PDE4D Q08499 1/20 0.35
ESR2 Q92731 1/20 0.34
GRM4 Q14833 1/20 0.33
FFAR1 O14842 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24629246 0.81 MAOB (0.43) GRM5
SCHEMBL24629247 0.77 KDM4E (0.38) GRM5
SCHEMBL24628992 0.76 PDE4B (0.41) PDE4D
SCHEMBL26895796 0.75 ESR2 (0.56) GRM5ESR2
SCHEMBL26854537 0.73 GRM5 (0.46) GRM5
SCHEMBL24628686 0.71 DRD2 (0.39) GRM5DRD2DRD1DRD4DRD5
SCHEMBL26895925 0.71 ALDH1A1 (0.46) PDE4D
SCHEMBL24628556 0.71 MEN1 (0.41) GRM5ESR2
SCHEMBL26896015 0.70 PRMT5 (0.37) ESR2DRD3
SCHEMBL11744257 0.68 ESR2 (0.54) PDE4DESR2DRD2DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022149617-A1 COMPOUND LIBRARY 中外製薬株式会社 2022-07-14 WO disclosed