SCHEMBL24628992

SCHEMBL24628992

O=Cc1ccc(C(=O)N2CCc3cc(O)cc(C#Cc4ccccc4)c3C2)o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.41
PDE4D Q08499 6/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26895925 0.84 ALDH1A1 (0.46) PDE4BPDE4DMAPTMEN1NPC1
SCHEMBL24628702 0.76 GRM5 (0.39) PDE4D
SCHEMBL26854537 0.75 GRM5 (0.46) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL26895796 0.73 ESR2 (0.56) MAPTMAPK1
SCHEMBL24629246 0.72 MAOB (0.43) MEN1ALDH1A1KMT2A
SCHEMBL24629247 0.69 KDM4E (0.38) MAPTNPC1ALDH1A1RAB9ATP53
SCHEMBL24628556 0.64 MEN1 (0.41) MAPTMEN1NPC1ALDH1A1POLB
SCHEMBL24628686 0.62 DRD2 (0.39)
SCHEMBL26896015 0.61 PRMT5 (0.37)
SCHEMBL4786676 0.60 PDE4B (0.77) PDE4BPDE4DABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022149617-A1 COMPOUND LIBRARY 中外製薬株式会社 2022-07-14 WO disclosed