SCHEMBL24680481

SCHEMBL24680481

CC(C)[C@@H](O)CNc1c(F)cc(Cl)cc1F

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.35
ADRA2B P18089 3/20 0.35
ADRA2C P18825 3/20 0.35
LMNA P02545 1/20 0.33
TRPV3 Q8NET8 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KCNH2 Q12809 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
ADRB1 P08588 3/20 0.32
ADRB3 P13945 3/20 0.32
ADRB2 P07550 2/20 0.32
ADRA1A P35348 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24680808 0.72 RAPGEF4 (0.42) LMNAKCNH2KDM4ETSHR
SCHEMBL24681373 0.67 SLC6A4 (0.36) ADRA2AADRA2BADRA2CSLC6A2SLC6A4
SCHEMBL3845491 0.67 TRPM5 (0.33)
SCHEMBL27248110 0.65 GABRA1 (0.38) KCNH2KDM4ETSHR
SCHEMBL4853844 0.64 THRB (0.41) CYP3A4KDM4E
SCHEMBL11196349 0.64 MMP2 (0.39) KDM4ETSHR
SCHEMBL11196347 0.64 MMP2 (0.39) KDM4ETSHR
SCHEMBL27995398 0.64 TSHR (0.35) SLC6A2SLC6A4KCNH2TSHR
SCHEMBL30850043 0.63 TRPV3 (0.44) TRPV3
SCHEMBL20542077 0.62 SMN1; SMN2 (0.37) LMNAKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022226667-A1 SUBSTITUTED AMINO PYRIDINE COMPOUNDS AS INHIBITORS OF THE HAEMATOPOIETIC PROGENITOR KINASE 1 (HPK1) ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR) (CA) 2022-11-03 WO disclosed