SCHEMBL2468236

SCHEMBL2468236

CCCNCCc1ccc(NS(=O)(=O)c2ccc(C(C)C)cc2)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.48
ADRB1 P08588 4/20 0.48
ADRB3 P13945 4/20 0.48
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
POLB P06746 1/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
KCNH2 Q12809 1/20 0.41
TRIM24 O15164 1/20 0.41
BRD1 O95696 1/20 0.41
BRPF1 P55201 1/20 0.41
PGR P06401 1/20 0.40
KIT P10721 1/20 0.40
GHSR Q92847 1/20 0.40
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4925564 0.99 ADRB2 (0.47) ADRB2ADRB1ADRB3ALDH1A1LMNA
SCHEMBL2470506 0.84 RAB9A (0.47) ADRB2ADRB1ADRB3ALDH1A1LMNA
SCHEMBL2470231 0.83 ALDH1A1 (0.47) ADRB2ADRB1ADRB3ALDH1A1LMNA
SCHEMBL1032588 0.82 MEN1 (0.43) ADRB2ADRB1ADRB3ALDH1A1LMNA
SCHEMBL2472514 0.82 ADRB2 (0.60) ADRB2ADRB1ADRB3ALDH1A1LMNA
Hydrochloric Acid SCHEMBL4244246 0.81 ADRB2 (0.42) ADRB2ADRB1ADRB3ALDH1A1LMNA
Hydrochloric Acid SCHEMBL4922779 0.81 ADRB2 (0.59) ADRB2ADRB1ADRB3ALDH1A1LMNA
SCHEMBL2468223 0.78 LMNA (0.46) ADRB2ADRB1ADRB3ALDH1A1LMNA
SCHEMBL1546730 0.71 DRD2 (0.49) ALDH1A1LMNAMAPTPKMSMN1; SMN2
SCHEMBL1032844 0.70 MEN1 (0.42) ADRB2ADRB1ADRB3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371814-A1 Aminoethylaromatic compounds suitable for treating disorders that respond to modulation of the dopamine D3 receptor Abbott GmbH & Co. KG (DE) 2011-10-05 EP disclosed
EP-1809597-A1 AMINOETHYLAROMATIC COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR Abbott GmbH & Co. KG (DE) 2007-07-25 EP disclosed
WO-2006040179-A1 AMINOETHYLAROMATIC COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR ABBOTT GMBH & CO. KG (DE) 2006-04-20 WO disclosed