SCHEMBL24716092

SCHEMBL24716092

CNC(=O)OCc1ccc(OC(C)=O)cc1C#N

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
AR P10275 1/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 2/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
CUL4A Q13619 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PKM P14618 1/20 0.35
LMNA P02545 2/20 0.35
ACHE P22303 1/20 0.35
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21728056 0.80 LMNA (0.43) CYP3A4NPC1RAB9AARTDP1
SCHEMBL24716090 0.80 MAOB (0.44) CYP3A4KDM4EMAPTMAPK1ALDH1A1
SCHEMBL24716095 0.76 EPHX2 (0.43) CYP3A4KDM4E
SCHEMBL24716093 0.75 CFD (0.42) CYP3A4KDM4EMAPTALDH1A1CYP1A2
SCHEMBL12863749 0.74 TOP2A (0.52) MAPTALDH1A1PKMLMNACYP1A2
SCHEMBL5263668 0.72 ACHE (0.54) CYP3A4ARTDP1KDM4EMAPT
SCHEMBL5630201 0.72 CYP3A4 (0.47) CYP3A4ARTDP1KDM4EMAPT
SCHEMBL28397412 0.71 LMNA (0.43) CYP3A4ARTDP1KDM4EMAPT
SCHEMBL28068682 0.71 MRGPRX4 (0.48) CYP3A4ARTDP1KDM4EMAPT
SCHEMBL18973312 0.70 RAB9A (0.48) CYP3A4NPC1RAB9ACASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022245759-A2 AGENTS FOR DIRECTED CONJUGATION TECHNIQUES AND CONJUGATED PRODUCTS BIOHAVEN THERAPEUTICS LTD. (US) 2022-11-24 WO disclosed