SCHEMBL24734855

SCHEMBL24734855

COc1ccc(OC)c2c1CCC(N)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 1.00
DRD2 P14416 2/20 0.65
DRD3 P35462 2/20 0.65
CYP1A2 P05177 1/20 0.45
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
PLAU P00749 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8669188 0.98 ADRA1A (0.96) ADRA1ADRD2DRD3CYP1A2HTR1D
Bromide SCHEMBL25243558 0.98 ADRA1A (0.96) ADRA1ADRD2DRD3CYP1A2HTR1D
Hydrochloric Acid SCHEMBL30861222 0.98 ADRA1A (0.96) ADRA1ADRD2DRD3CYP1A2HTR1D
SCHEMBL7551749 0.89 ADRA1A (0.79) ADRA1ADRD2DRD3CYP1A2
SCHEMBL4217393 0.88 ADRA1A (0.78) ADRA1ADRD2DRD3CYP1A2
SCHEMBL7549300 0.88 ADRA1A (0.78) ADRA1ADRD2DRD3CYP1A2
SCHEMBL5793364 0.88 ADRA1A (0.78) ADRA1ADRD2DRD3CYP1A2HTR1D
SCHEMBL7245131 0.88 ADRA1A (0.78) ADRA1ADRD2DRD3CYP1A2HTR1D
SCHEMBL7028738 0.88 ADRA1A (0.78) ADRA1ADRD2DRD3CYP1A2HTR1D
SCHEMBL7028736 0.88 ADRA1A (0.78) ADRA1ADRD2DRD3CYP1A2HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250282708-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI THERAPEUTICS, INC. (US) 2025-09-11 US claimed
US-12344570-B2 Aminotetraline activators of serotonin receptors ATAI THERAPEUTICS, INC. (US) 2025-07-01 US claimed
EP-4457203-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI Therapeutics, Inc. (US) 2024-11-06 EP claimed
US-20240300885-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI Life Sciences AG (DE) 2024-09-12 US claimed
US-11827580-B2 Aminotetraline activators of serotonin receptors ATAI Life Sciences AG (DE) 2023-11-28 US claimed
WO-2023129909-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI Life Sciences AG (DE) 2023-07-06 WO claimed
US-20230202965-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ENTHEOGENIX BIOSCIENCES, INC. 2023-06-29 US claimed
US-20250282708-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI THERAPEUTICS, INC. (US) 2025-09-11 US disclosed
US-12344570-B2 Aminotetraline activators of serotonin receptors ATAI THERAPEUTICS, INC. (US) 2025-07-01 US disclosed
EP-4457203-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI Therapeutics, Inc. (US) 2024-11-06 EP disclosed
US-20240300885-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI Life Sciences AG (DE) 2024-09-12 US disclosed
US-11827580-B2 Aminotetraline activators of serotonin receptors ATAI Life Sciences AG (DE) 2023-11-28 US disclosed
US-11827580-B2 Aminotetraline activators of serotonin receptors ATAI Life Sciences AG (DE) 2023-11-28 US disclosed
WO-2023129909-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI Life Sciences AG (DE) 2023-07-06 WO disclosed
US-20230202965-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ENTHEOGENIX BIOSCIENCES, INC. 2023-06-29 US disclosed
US-20230202965-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ENTHEOGENIX BIOSCIENCES, INC. 2023-06-29 US disclosed
US-20230202965-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS ENTHEOGENIX BIOSCIENCES, INC. 2023-06-29 US disclosed
US-20230138118-A1 DIMETHOXYPHENYLALKYLAMINE ACTIVATORS OF SEROTONIN RECEPTORS Atai Therapeutics Inc. 2023-05-04 US disclosed
US-20230138118-A1 DIMETHOXYPHENYLALKYLAMINE ACTIVATORS OF SEROTONIN RECEPTORS Atai Therapeutics Inc. 2023-05-04 US disclosed
WO-2022261240-A2 DIMETHOXYPHENYLALKYLAMINE ACTIVATORS OF SEROTONIN RECEPTORS ATAI Life Sciences AG (DE) 2022-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240300885-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS HTR3B, HTR1B, TAAR5 ADRA1A 32/4885DRD2 111/4885DRD3 273/4885
US-20230138118-A1 DIMETHOXYPHENYLALKYLAMINE ACTIVATORS OF SEROTONIN RECEPTORS HTR1A, HTR7, HTR4 ADRA1A 23/4885DRD2 25/4885DRD3 57/4885
US-20250282708-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS HTR3B, HTR1B, TAAR5 ADRA1A 32/4885DRD2 111/4885DRD3 273/4885
US-12344570-B2 Aminotetraline activators of serotonin receptors HTR3B, HTR1B, TAAR5 ADRA1A 32/4885DRD2 111/4885DRD3 273/4885
US-11827580-B2 Aminotetraline activators of serotonin receptors HTR3B, HTR1B, TAAR5 ADRA1A 28/4885DRD2 98/4885DRD3 266/4885
US-20230202965-A1 AMINOTETRALINE ACTIVATORS OF SEROTONIN RECEPTORS HTR3B, HTR1B, TAAR5 ADRA1A 32/4885DRD2 111/4885DRD3 273/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.