SCHEMBL2474145

SCHEMBL2474145

CCCC[Sn](CCCC)(CCCC)c1nc2ccccc2o1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPT P10636 4/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
ALDH1A1 P00352 2/20 0.43
KMT2A Q03164 2/20 0.43
HSD17B10 Q99714 2/20 0.43
LMNA P02545 2/20 0.43
F2 P00734 1/20 0.43
MIF P14174 1/20 0.43
TP53 P04637 3/20 0.41
FAAH O00519 2/20 0.41
CES1 P23141 1/20 0.41
HSP90AA1 P07900 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
PTGS2 P35354 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4261648 0.83 NPC1 (0.48) TDP1MAPTNPC1RAB9AALDH1A1
SCHEMBL6418155 0.82 ATM (0.41) ATMTDP1L3MBTL1MAPTNPC1
SCHEMBL591905 0.71 RAB9A (0.72) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL30184671 0.71 RAB9A (0.72) MAPTNPC1RAB9AALDH1A1KMT2A
Benzene SCHEMBL28280876 0.70 RAB9A (0.70) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL439174 0.70 MAPT (0.70) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL2567453 0.69 MAPT (0.68) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL14402606 0.69 MAPT (0.68) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL7793708 0.69 MAPT (0.68) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL11623669 0.69 MAPT (0.68) MAPTNPC1RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4539840-A1 KINASE MODULATORS AND METHODS OF USE THEREOF Neuron23, Inc. (US) 2025-04-23 EP disclosed
CN-119730846-A Kinase modulators and methods of use thereof 神经元23公司 2025-03-28 CN disclosed
WO-2023244788-A9 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. (US) 2024-09-12 WO disclosed
US-20240025906-A1 KINASE MODULATORS AND METHODS OF USE THEREOF SUNDANCE BIOSCIENCES, INC. 2024-01-25 US disclosed
WO-2023244788-A1 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. (US) 2023-12-21 WO disclosed
US-10640510-B2 Metabotrophic glutamate receptor 5 modulators and methods use thereof SUNOVION PHARMACEUTICALS INC. (US) 2020-05-05 US disclosed
US-20200079778-A9 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF SUNOVION PHARMACEUTICALS INC. 2020-03-12 US disclosed
US-20190135815-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2019-05-09 US disclosed
US-10196399-B2 Metabotrophic glutamate receptor 5 modulators and methods use thereof SUNOVION PHARMACEUTICALS INC. (US) 2019-02-05 US disclosed
US-20180037585-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF SUNOVION PHARAMCEUTICALS INC. 2018-02-08 US disclosed
EP-1390433-B1 SYNTHESIS AND EVALUATION OF NEW CYANINE DYES AS MINOR GROOVE OF POLY(DA-DT)] 2 BINDERS LIGHT UP TECHNOLOGIES AB (SE) 2005-02-16 EP disclosed
US-20040229910-A1 Therapeutic compounds N.V. ORGANON (NL) 2004-11-18 US disclosed
US-20040132046-A1 Synthesis and evaluation of new cyanine dyes as minor groove of [POLY (dA-dT)]2 binders LIGHT UP TECHNOLOGIES AB (SE) 2004-07-08 US disclosed
EP-1390433-A1 SYNTHESIS AND EVALUATION OF NEW CYANINE DYES AS MINOR GROOVE OF POLY(DA-DT)] 2 BINDERS Light Up Technologies AB (SE) 2004-02-25 EP disclosed
WO-2002090443-A1 SYNTHESIS AND EVALUATION OF NEW CYANINE DYES AS MINOR GROOVE OF [POLY(DA-DT)]2 BINDERS LIGHT UP TECHNOLOGIES AB (SE) 2002-11-14 WO disclosed
US-20020037885-A1 Therapeutic compounds DIJCKS FREDERICUS ANTONIUS (NL) 2002-03-28 US disclosed
US-6313139-B1 ADMINISTERING BENZYLAMINE DERIVATIVE FOR THERAPY OF PSYCHIATRIC DISORDER IN MAMMALS AKZO NOBEL N. V. (NL) 2001-11-06 US disclosed
EP-1035843-A2 I h?-MODULATORS Akzo Nobel N.V. (NL) 2000-09-20 EP disclosed
US-6080773-A USEFUL FOR TREATMENT OF DEPRESSION, ANXIETY OR PSYCHOSIS AKZO NOBEL, N.V. (NL) 2000-06-27 US disclosed
WO-1999018941-A2 Ih-MODULATORS AKZO NOBEL N.V. (NL) 1999-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10196399-B2 Metabotrophic glutamate receptor 5 modulators and methods use thereof GRM5, GRIK5, GRM2 ATM 4438/4885TDP1 3830/4885L3MBTL1 3852/4885
US-20040229910-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 ATM 2418/4885TDP1 2228/4885L3MBTL1 3374/4885
US-20180037585-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF GRM5, GRIK5, GRM2 ATM 4438/4885TDP1 3830/4885L3MBTL1 3852/4885
US-20190135815-A1 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF GRM5, GRIK5, GRM2 ATM 4438/4885TDP1 3830/4885L3MBTL1 3852/4885
US-20200079778-A9 METABOTROPHIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS USE THEREOF GRM5, GRIK5, GRM2 ATM 4438/4885TDP1 3830/4885L3MBTL1 3852/4885
US-10640510-B2 Metabotrophic glutamate receptor 5 modulators and methods use thereof GRM5, GRIK5, GRM2 ATM 4438/4885TDP1 3830/4885L3MBTL1 3852/4885
US-20020037885-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 ATM 2418/4885TDP1 2228/4885L3MBTL1 3374/4885
US-20240025906-A1 KINASE MODULATORS AND METHODS OF USE THEREOF TYK2, JAK1, JAK3 ATM 710/4885TDP1 1065/4885L3MBTL1 1224/4885
US-20040132046-A1 Synthesis and evaluation of new cyanine dyes as minor groove of [POLY (dA-dT)]2 binders DRD4, FUT4, DRD1 ATM 3844/4885TDP1 1639/4885L3MBTL1 3273/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.