SCHEMBL247492

SCHEMBL247492

Cc1cccc(CC=O)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
CCR1 P32246 1/20 0.43
CCR8 P51685 1/20 0.43
NOS3 P29474 1/20 0.40
NOS2 P35228 1/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
P2RX7 Q99572 1/20 0.39
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
RAB9A P51151 2/20 0.37
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
HPGD P15428 2/20 0.36
GRM5 P41594 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22482055 0.84 PGK1 (0.43) NOS2NPSR1
SCHEMBL2010535 0.81 CCR1 (0.44) SMN1; SMN2CCR1CCR8NOS3NOS2
SCHEMBL943326 0.80
SCHEMBL6193822 0.80 SMN1; SMN2 (0.45) SMN1; SMN2CCR1CCR8NOS3NOS2
SCHEMBL17429701 0.79 CCR1 (0.43) SMN1; SMN2CCR1CCR8NOS3NOS2
SCHEMBL13879249 0.78 NOS2 (0.43) SMN1; SMN2CCR1CCR8NOS3NOS2
SCHEMBL6195640 0.77 KCNH2 (0.43) SMN1; SMN2CCR1CCR8NOS3NOS2
SCHEMBL24259223 0.76 KCNH2 (0.46) SMN1; SMN2CCR1CCR8NOS3NOS2
SCHEMBL243243 0.76
SCHEMBL20730061 0.75 PGK1 (0.41) CCR1NPSR1MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4514802-A1 IMIDAZOLE DERIVATIVES AS ALK5 INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2025-03-05 EP disclosed
WO-2023247592-A1 5-(4-FLUOROPHENYL)-2,3-DIHYDRO-1H-IMIDAZO[1,2-A]IMIDAZOLE DERIVATIVES AS ALK INHIBITORS FOR THE TREATMENT OF FIBROSIS CHIESI FARMACEUTICI S.P.A. (IT) 2023-12-28 WO disclosed
WO-2023208986-A1 IMIDAZOLE DERIVATIVES AS ALK5 INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2023-11-02 WO disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-11471867-B2 Ligand for forming ruthenium complex, ruthenium complex catalyst, production method therefor and use thereof GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2022-10-18 US disclosed
WO-2022076905-A1 ALK5 INHIBITORS, CONJUGATES, AND USES THEREOF SILVERBACK THERAPEUTICS, INC. (US) 2022-04-14 WO disclosed
EP-3820474-A1 ADENOSINE RECEPTOR BINDING COMPOUNDS Nikang Therapeutics, Inc. (US) 2021-05-19 EP disclosed
EP-3774782-A2 ATF6 INHIBITORS AND USES THEREOF Black Belt TX Ltd (GB) 2021-02-17 EP disclosed
US-20200360911-A1 LIGAND FOR FORMING RUTHENIUM COMPLEX, RUTHENIUM COMPLEX CATALYST, PRODUCTION METHOD THEREFOR AND USE THEREOF GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2020-11-19 US disclosed
EP-3057948-A1 SELECTIVELY SUBSTITUTED QUINOLINE COMPOUNDS Eisai R&D Management Co., Ltd. (JP) 2016-08-24 EP disclosed
WO-2008074418-A2 BISOXIMES AS FUNGICIDES AND ARTHROPODICIDES BAYER CROPSCIENCE AKTENGESELLSCHAFT (DE) 2008-06-26 WO disclosed
US-7087626-B2 Pyrrole derivatives as pharmaceutical agents ELI LILLY AND COMPANY (US) 2006-08-08 US disclosed
EP-1601676-A2 FUSED IMIDAZOLES AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS Pfizer Products Inc. (US) 2005-12-07 EP disclosed
EP-1542994-A1 NOVEL TRIAZOLE AND OXAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITOR Pfizer Products Inc. (US) 2005-06-22 EP disclosed
EP-1542684-A2 NOVEL PYRAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS Pfizer Products Inc. (US) 2005-06-22 EP disclosed
WO-2004078110-A2 FUSED IMIZADOLES AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS PFIZER PRODUCTS INC. (US) 2004-09-16 WO disclosed
WO-2004026863-A1 NOVEL OXAZOLE AND THIAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS PFIZER PRODUCTS INC. (US) 2004-04-01 WO disclosed
WO-2004026306-A2 PYRAZOLE DERIVATIVES AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS PFIZER PRODUCTS INC. (US) 2004-04-01 WO disclosed
EP-0974602-B1 Catalyst and process for hydrogenating olefinically unsaturated compound JSR CORP (JP) 2004-01-02 EP disclosed
CN-1281436-A N-Benzyl-3-indenylacetamides derivatives for treating neoplasia CELL PATHWAYS INC (US) 2001-01-24 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133132-A1 NAMPT MODULATORS NAMPT, MC4R, SIRT1 SMN1; SMN2 1161/4885CCR1 4148/4885CCR8 4238/4885
US-11471867-B2 Ligand for forming ruthenium complex, ruthenium complex catalyst, production method therefor and use thereof NOTUM, WEE2, WEE1 SMN1; SMN2 4861/4885CCR1 2048/4885CCR8 1824/4885
US-20200360911-A1 LIGAND FOR FORMING RUTHENIUM COMPLEX, RUTHENIUM COMPLEX CATALYST, PRODUCTION METHOD THEREFOR AND USE THEREOF NOTUM, WEE2, WEE1 SMN1; SMN2 4861/4885CCR1 2048/4885CCR8 1824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.