SCHEMBL2482791

SCHEMBL2482791

CC1=C[CH]CC=C1N1CCN(CC2CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.34
CASP4 P49662 1/20 0.34
CASP5 P51878 1/20 0.34
DRD2 P14416 2/20 0.33
DRD3 P35462 1/20 0.33
KDM2B Q8NHM5 2/20 0.32
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2485210 0.76 KMT2A (0.33)
SCHEMBL2483016 0.74 GPR119 (0.30)
SCHEMBL2477477 0.69 NPSR1 (0.43)
SCHEMBL2483385 0.69 CASP1 (0.35) CASP1CASP4CASP5DRD2DRD3
SCHEMBL12082219 0.66 MAPT (0.51) DRD2DRD3
SCHEMBL18740713 0.65
SCHEMBL7321483 0.65 CHRM5 (0.60) CASP1CASP4CASP5DRD2ACHE
Hydrochloric Acid SCHEMBL7331633 0.63 CHRM5 (0.57) ACHE
SCHEMBL15499062 0.61 MAPT (0.47) DRD2DRD3ACHE
SCHEMBL11084741 0.61 DRD2 (0.67) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376494-A1 DIHYDROPYRIMIDOPYRIMIDINE DERIVATIVES MSD K.K. (JP) 2011-10-19 EP disclosed
EP-2376493-A1 DIHYDROPYRIMIDOPYRIMIDINE DERIVATIVE MSD K.K. (JP) 2011-10-19 EP disclosed
WO-2010067886-A1 DIHYDROPYRIMIDOPYRIMIDINE DERIVATIVE BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-06-17 WO disclosed
WO-2010067888-A1 DIHYDROPYRIMIDOPYRIMIDINE DERIVATIVES BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-06-17 WO disclosed