SCHEMBL2487330

SCHEMBL2487330

CC(C)(C)C(C(=O)O)n1ccc2cc(C#N)ccc21.CC(C)(C)OC(=O)CBr

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.36
ABCB1 P08183 9/20 0.36
CCR9 P51686 2/20 0.34
NR1H2 P55055 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
NTRK1 P04629 1/20 0.32
NPY5R Q15761 1/20 0.32
HTR6 P50406 2/20 0.31
DRD2 P14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2414232 0.87 CCR9 (0.39) FFAR4ABCB1CCR9IRAK4NTRK1
SCHEMBL3467553 0.81 KDM4E (0.41) FFAR4ABCB1NPY5R
SCHEMBL27844158 0.74 NPY5R (0.45) FFAR4ABCB1CCR9NPY5R
SCHEMBL7367610 0.72 FFAR4 (0.41) FFAR4ABCB1CCR9IRAK4NPY5R
SCHEMBL1876083 0.70 PIK3CD (0.44) FFAR4CCR9NR1H2IRAK4HTR6
SCHEMBL1435781 0.66 NPY5R (0.42) ABCB1IRAK4NPY5RDRD2
SCHEMBL2951656 0.66 DRD2 (0.40) FFAR4ABCB1NPY5RHTR6DRD2
SCHEMBL1435785 0.66 NPY5R (0.42) ABCB1IRAK4NPY5RDRD2
SCHEMBL3709688 0.66 CDC7 (0.43) FFAR4NPY5RHTR6
SCHEMBL9009161 0.65 MTNR1A (0.47) NPY5RDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376484-A1 OXADIAZOLE FUSED HETEROCYCLIC DERIVATIVES USEFUL FOR THE TREATMENT OF MULTIPLE SCLEROSIS Merck Serono S.A. (CH) 2011-10-19 EP disclosed