SCHEMBL2491318

SCHEMBL2491318

CNc1ccc(-c2ccc(Cn3cc(OC(=O)O)c(=O)c4c(NC)cccc43)cc2)cn1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.40
TOP1 P11387 3/20 0.37
TP53 P04637 3/20 0.35
CNR2 P34972 1/20 0.35
MAPT P10636 1/20 0.35
LMNA P02545 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487138 0.90 CHRM1 (0.52) CHRM1TOP1TP53CNR2
SCHEMBL2485890 0.86 CHRM1 (0.56) CHRM1TOP1LMNA
SCHEMBL2490909 0.79 CHRM1 (0.50) CHRM1TOP1TP53
SCHEMBL2489733 0.78 CHRM1 (0.57) CHRM1TOP1TP53CNR2LMNA
SCHEMBL2487134 0.76 CHRM1 (0.71) CHRM1TOP1TP53LMNA
SCHEMBL2490524 0.74 CHRM1 (0.71) CHRM1TOP1TP53CNR2LMNA
SCHEMBL2487860 0.72 CNR2 (0.41) CHRM1CNR2MAPT
SCHEMBL2490511 0.72 LMNA (0.59) CHRM1TP53CNR2LMNA
SCHEMBL2489217 0.72 CHRM1 (0.61) CHRM1TP53LMNA
SCHEMBL2491670 0.71 CHRM1 (0.52) CHRM1TOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2037739-B1 BENZYL-SUBSTITUTED QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2011-10-26 EP claimed