SCHEMBL24920403

SCHEMBL24920403

COc1cnnc(-n2nccn2)c1

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.32
HCRTR2 O43614 2/20 0.32
ALDH1A1 P00352 1/20 0.31
ROCK2 O75116 1/20 0.31
MAP4K4 O95819 1/20 0.31
PRKACA P17612 1/20 0.31
ROCK1 Q13464 1/20 0.31
DYRK1A Q13627 1/20 0.31
NTRK3 Q16288 1/20 0.31
PKN2 Q16513 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
STK17A Q9UEE5 1/20 0.31
CCR1 P32246 1/20 0.31
CCR5 P51681 1/20 0.31
CCR8 P51685 1/20 0.31
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920809 0.81 PDE10A (0.34)
SCHEMBL24920821 0.76 KDM4E (0.43) ALDH1A1NOTUM
SCHEMBL24920393 0.72 CCR1 (0.53) HCRTR1HCRTR2ROCK1DYRK1ACLK4
SCHEMBL24920899 0.71 TDO2 (0.36)
SCHEMBL24920389 0.69 GABRG2 (0.38) HCRTR1HCRTR2ALDH1A1
SCHEMBL14982162 0.69 ADRB1 (0.51)
SCHEMBL24921192 0.68 CHRNB2 (0.49) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL20912238 0.68 EGLN1 (0.39) HCRTR1HCRTR2ALDH1A1CLK4CCR1
SCHEMBL2614481 0.67
SCHEMBL19480834 0.67 HCRTR1 (0.37) HCRTR1HCRTR2ALDH1A1ROCK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed