SCHEMBL24933726

SCHEMBL24933726

C=C(Nc1cccc(C)c1)c1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.54
BRAF P15056 1/20 0.51
KCNK3 O14649 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
CSF1R P07333 1/20 0.49
HTT P42858 2/20 0.49
GAA P10253 2/20 0.49
ALDH1A1 P00352 1/20 0.49
KMT2A Q03164 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 2/20 0.49
PKM P14618 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
IMPDH2 P12268 1/20 0.48
TSHR P16473 1/20 0.48
RAB9A P51151 1/20 0.48
KCNK9 Q9NPC2 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL259177 0.82 TDP1 (0.78) TDP1BRAFKCNK3CYP1A2CYP2C9
SCHEMBL12707417 0.81 MEN1 (0.57) TDP1KCNK3CYP1A2CYP3A4CYP2C9
SCHEMBL19608697 0.76 GAA (0.51) TDP1CYP1A2CYP3A4CYP2C19GAA
SCHEMBL9192069 0.76 KMT2A (0.72) BRAFCYP1A2HTTGAAALDH1A1
Hydrochloric Acid SCHEMBL9187992 0.75 KMT2A (0.70) BRAFCYP1A2HTTGAAALDH1A1
SCHEMBL9435155 0.74 TDP1 (0.62) TDP1BRAFKCNK3CYP1A2CYP3A4
SCHEMBL2790141 0.74 KMT2A (0.67) TDP1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5214513 0.74 TDP1 (0.57) TDP1BRAFKCNK3CYP1A2CYP3A4
SCHEMBL25872256 0.74 ALDH1A1 (0.55) KCNK3CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL31661935 0.73 BRAF (0.79) TDP1BRAFKCNK3CSF1RALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023009475-A1 ROCK2 INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-02-02 WO disclosed