SCHEMBL2493594

SCHEMBL2493594

CC(=Nc1ccc(Cl)nn1)N(C)C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
USP2 O75604 1/20 0.34
RECQL P46063 1/20 0.34
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15562694 1.00 ALDH1A1 (0.34) ALDH1A1USP2RECQLNPC1RAB9A
SCHEMBL2493593 1.00 ALDH1A1 (0.34) ALDH1A1USP2RECQLNPC1RAB9A
SCHEMBL6219536 0.83 ALDH1A1 (0.35) ALDH1A1USP2RECQLGAAMAPT
SCHEMBL6213276 0.79 NOS1 (0.38) ALDH1A1USP2RECQLGAAMAPT
SCHEMBL6213273 0.79 NOS1 (0.38) ALDH1A1USP2RECQLGAAMAPT
SCHEMBL16792283 0.78
SCHEMBL18339066 0.78
SCHEMBL6621084 0.77 LMNA (0.33) ALDH1A1USP2RECQL
SCHEMBL6279198 0.77 USP2 (0.32) ALDH1A1USP2RECQL
SCHEMBL6279200 0.77 USP2 (0.32) ALDH1A1USP2RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4709722-A1 ISOXAZOLIDINES AS RIPK1 INHIBITORS AND USE THEREOF GENZYME CORPORATION (US) 2026-03-18 EP disclosed
WO-2024233547-A1 ISOXAZOLIDINES AS RIPK1 INHIBITORS AND USE THEREOF GENZYME CORPORATION (US) 2024-11-14 WO disclosed
EP-3080128-B1 IMIDAZOPYRIDAZINE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB Biopharma SRL (BE) 2020-06-24 EP disclosed
EP-3298017-B1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY HOFFMANN LA ROCHE (CH) 2019-08-14 EP disclosed
US-10208067-B2 Compounds for treating spinal muscular atrophy HOFFMANN-LA ROCHE INC. (US) 2019-02-19 US disclosed
US-20180194781-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY HOFFMANN-LA ROCHE INC. (US) 2018-07-12 US disclosed
EP-3298017-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY H. Hoffnabb-La Roche Ag (CH) 2018-03-28 EP disclosed
US-9873703-B2 Imidazopyridazine derivatives as modulators of TNF activity UCB BIOPHARMA SPRL (BE) 2018-01-23 US disclosed
US-20160376275-A1 Imidazopyridazine Derivatives as Modulators of TNF Activity UCB BIOPHARMA SPRL (BE) 2016-12-29 US disclosed
WO-2016184832-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY F. HOFFMANN-LA ROCHE AG (CH) 2016-11-24 WO disclosed
WO-2014020531-A1 IMIDAZO[1,2-B]PYRIDAZIN-6-AMINE DERIVATIVES AS KINASE JAK-2 INHIBITORS CELON PHARMA S.A. (PL) 2014-02-06 WO disclosed
EP-2379557-B1 AMINO PYRAZOLE COMPOUND LILLY CO ELI (US) 2012-10-31 EP disclosed
EP-2379557-A1 AMINO PYRAZOLE COMPOUND Eli Lilly and Company (US) 2011-10-26 EP disclosed
US-7897600-B2 Amino pyrazole compound ELI LILLY AND COMPANY (US) 2011-03-01 US disclosed
US-20100286139-A1 AMINO PYRAZOLE COMPOUND ELI LILLY AND COMPANY (US) 2010-11-11 US disclosed
WO-2010074947-A1 AMINO PYRAZOLE COMPOUND ELI LILLY AND COMPANY (US) 2010-07-01 WO disclosed
US-20100152181-A1 AMINO PYRAZOLE COMPOUND ELI LILLY AND COMPANY (US) 2010-06-17 US disclosed
EP-1362050-B1 PYRIMIDINE DERIVATIVES FOR INHIBITION OF CELL-PROLIFERATION ASTRAZENECA AB (SE) 2005-02-02 EP disclosed
US-6844341-B2 Pyrimidine derivatives for inhibition of cell proliferation ASTRAZENECA AB (SE) 2005-01-18 US disclosed
US-20040097506-A1 Pyrimidine derivatives for inhibition of cell proliferation ASTRAZENECA AB (SE) 2004-05-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160376275-A1 Imidazopyridazine Derivatives as Modulators of TNF Activity TNF, TNFRSF1A, IL1A ALDH1A1 217/4885USP2 3509/4885RECQL 1878/4885
US-20040097506-A1 Pyrimidine derivatives for inhibition of cell proliferation TYMP, TK1, TYMS ALDH1A1 127/4885USP2 4225/4885RECQL 23/4885
US-20100286139-A1 AMINO PYRAZOLE COMPOUND MCL1, MYC, PML ALDH1A1 2620/4885USP2 3065/4885RECQL 4807/4885
US-20180194781-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, PYGM, CPT1B ALDH1A1 770/4885USP2 2940/4885RECQL 135/4885
US-20100152181-A1 AMINO PYRAZOLE COMPOUND MCL1, MYC, PML ALDH1A1 2620/4885USP2 3065/4885RECQL 4807/4885
US-10208067-B2 Compounds for treating spinal muscular atrophy SMN1; SMN2, PYGM, CPT1B ALDH1A1 770/4885USP2 2940/4885RECQL 135/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.