SCHEMBL24959136

SCHEMBL24959136

OCc1ncc(C(F)(F)F)s1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPM5 Q9NZQ8 1/20 0.41
FFAR2 O15552 2/20 0.34
MLYCD O95822 2/20 0.32
TRPV1 Q8NER1 1/20 0.31
DAO P14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2469989 0.82 MLYCD (0.46) MLYCD
SCHEMBL20098867 0.81 TRPM5 (0.42) TRPM5FFAR2MLYCD
SCHEMBL24958959 0.79 TRPM5 (0.41) TRPM5FFAR2
SCHEMBL17018480 0.76 LOXL2 (0.32)
SCHEMBL10965044 0.72 TRPM5 (0.35) TRPM5
SCHEMBL7252403 0.72 ALDH1A1 (0.42) TRPM5MLYCD
SCHEMBL25145638 0.69 CACNA1H (0.42) TRPM5
SCHEMBL31078390 0.69 ALDH1A1 (0.34) TRPM5FFAR2MLYCDDAO
SCHEMBL2956791 0.69
SCHEMBL27323915 0.68 ALDH1A1 (0.39) TRPM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117295729-A Carboxy-benzimidazole GLP-1R modulating compounds 吉利德科学公司 2023-12-26 CN disclosed
EP-4271674-A1 CARBOXY-BENZIMIDAZOLE GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-11-08 EP disclosed
US-20230021705-A1 GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-01-26 US disclosed
WO-2022225914-A1 CARBOXY-BENZIMIDAZOLE GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-10-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230021705-A1 GLP-1R MODULATING COMPOUNDS GLP1R, GIPR, GPR119 TRPM5 1457/4885FFAR2 78/4885MLYCD 1403/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.