SCHEMBL24967931

SCHEMBL24967931

COC(=O)Cc1cccc(-c2cnc(OC)c(C(F)(F)F)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 3/20 0.55
LMNA P02545 1/20 0.47
CDK8 P49336 2/20 0.45
PIK3CD O00329 4/20 0.45
PIK3CG P48736 3/20 0.45
PIK3CA P42336 2/20 0.45
PIK3CB P42338 2/20 0.45
KCNH2 Q12809 1/20 0.45
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
AAK1 Q2M2I8 1/20 0.41
VEGFA P15692 1/20 0.40
FLT1 P17948 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
EGLN3 Q9H6Z9 1/20 0.40
GRIN1 Q05586 2/20 0.39
GRIN2B Q13224 2/20 0.39
NR1H2 P55055 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30851237 0.90 NR1H2 (0.48) SYKCDK8PIK3CDPIK3CGPIK3CA
SCHEMBL24967930 0.90 NR1H2 (0.48) SYKCDK8PIK3CDPIK3CGPIK3CA
SCHEMBL24967940 0.78 HSD17B1 (0.52) SYKPIK3CDPIK3CGPIK3CAPIK3CB
SCHEMBL30851292 0.78 HSD17B1 (0.52) SYKPIK3CDPIK3CGPIK3CAPIK3CB
SCHEMBL24967932 0.77 PIK3CD (0.48) SYKLMNACDK8PIK3CDPIK3CG
SCHEMBL30165044 0.77 PIK3CD (0.48) SYKLMNACDK8PIK3CDPIK3CG
SCHEMBL21915788 0.76 LMNA (0.50) SYKLMNANR1H2NR1H3POLB
SCHEMBL6270689 0.75 AGXT (0.56) SYKNR1H2NR1H3POLBSLC7A5
SCHEMBL3933089 0.74 ALDH1A1 (0.60) SYKCYP11B1CYP11B2SLC7A5KDM4E
SCHEMBL3930818 0.74 MAP4K4 (0.57) SYKCYP11B1CYP11B2CYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117642393-A Novel PARP7 inhibitor and application thereof 上海齐鲁制药研究中心有限公司 2024-03-01 CN disclosed
WO-2023006013-A1 NOVEL PARP7 INHIBITOR AND USE THEREOF 上海齐鲁制药研究中心有限公司 2023-02-02 WO disclosed