SCHEMBL25076280

SCHEMBL25076280

NC1CCOC(C2c3ccccc3CCc3ccccc32)C1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.39
RET P07949 1/20 0.39
SIGMAR1 Q99720 3/20 0.38
IDO1 P14902 4/20 0.37
PLAU P00749 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25076342 1.00 HTR2A (0.39) HTR2ARETSIGMAR1IDO1PLAU
SCHEMBL25076345 1.00 HTR2A (0.39) HTR2ARETSIGMAR1IDO1PLAU
SCHEMBL25076414 0.81 SIGMAR1 (0.41) HTR2ARETSIGMAR1
SCHEMBL25076434 0.80 KDM1A (0.33) HTR2AIDO1
SCHEMBL25076290 0.76 SIGMAR1 (0.41) HTR2ARETSIGMAR1IDO1
SCHEMBL25076341 0.75 SIGMAR1 (0.33) HTR2ARETSIGMAR1
SCHEMBL18045643 0.74 HTR2A (0.45) HTR2ARETSIGMAR1IDO1
SCHEMBL30096678 0.74 HTR2A (0.45) HTR2ARETSIGMAR1IDO1
SCHEMBL23832807 0.74 HTR2A (0.45) HTR2ARETSIGMAR1IDO1
SCHEMBL25761550 0.73 MTNR1A (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260062397-A1 2-DIARYLMETHYL-4-AMINOTETRAHYDROPYRAN DERIVATIVES AND RELATED COMPOUNDS AS ANTICANCER, ANTIINFLAMMATORY, ANTIFIBROTIC AND NEUROPROTECTIVE AGENTS ATUX ISKAY LLC (US) 2026-03-05 US disclosed
US-12522575-B2 2-diarylmethyl-4-aminotetrahydropyran derivatives and related compounds as anticancer, antiinflammatory, antifibrotic and neuroprotective agents ATUX ISKAY LLC (US) 2026-01-13 US disclosed
US-20250376455-A1 2-DIARYLMETHYL-4-AMINOTETRAHYDROPYRAN DERIVATIVES AND RELATED COMPOUNDS AS ANTICANCER, ANTIINFLAMMATORY, ANTIFIBROTIC AND NEUROPROTECTIVE AGENTS ATUX ISKAY LLC (US) 2025-12-11 US disclosed
WO-2023023594-A9 2‑DIARYLMETHYL‑4‑AMINOTETRAHYDROPYRAN DERIVATIVES AND RELATED COMPOUNDS AS ANTICANCER, ANTIINFLAMMATORY, ANTIFIBROTIC AND NEUROPROTECTIVE AGENTS ATUX ISKAY LLC (US) 2023-06-08 WO disclosed
WO-2023023594-A1 2‑DIARYLMETHYL‑4‑AMINOTETRAHYDROPYRAN DERIVATIVES AND RELATED COMPOUNDS AS ANTICANCER, ANTIINFLAMMATORY, ANTIFIBROTIC AND NEUROPROTECTIVE AGENTS ATUX ISKAY LLC (US) 2023-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250376455-A1 2-DIARYLMETHYL-4-AMINOTETRAHYDROPYRAN DERIVATIVES AND RELATED COMPOUNDS AS ANTICANCER, ANTIINFLAMMATORY, ANTIFIBROTIC AND NEUROPROTECTIVE AGENTS MYC, MYCBP, MYCBP2 HTR2A 2541/4885RET 2732/4885SIGMAR1 4024/4885
US-20260062397-A1 2-DIARYLMETHYL-4-AMINOTETRAHYDROPYRAN DERIVATIVES AND RELATED COMPOUNDS AS ANTICANCER, ANTIINFLAMMATORY, ANTIFIBROTIC AND NEUROPROTECTIVE AGENTS MYC, MYCBP, FOXO1 HTR2A 2108/4885RET 2220/4885SIGMAR1 3290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.