SCHEMBL2519264

SCHEMBL2519264

C1=CC(C2NCC23CCNCC3)c2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2436751 0.69 PRCP (0.39) HTR2CHTR2B
SCHEMBL5698322 0.68 HTR2A (0.44) HTR2CHTR2B
SCHEMBL2519261 0.64 TSHR (0.44) HTR2CHTR2B
SCHEMBL10352714 0.63 HTR2A (0.38) HTR2CHTR2B
SCHEMBL15571073 0.62 SIGMAR1 (0.42) OPRM1OPRD1
SCHEMBL30790640 0.62 HTR6 (0.33)
SCHEMBL1074094 0.61 HTR2A (0.35) HTR2CHTR2B
SCHEMBL7185808 0.61 HTR2A (0.35)
SCHEMBL28839778 0.61 HTR2A (0.35)
SCHEMBL7185802 0.61 HTR2A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547679-A1 2,3 DIHYDRO-1H-INDEN-1-YL- 2,7-DIAZASPIRO [3.6]NONANE DERIVATIVES AND THEIR USE AS ANTAGONISTS OR INVERSE AGONISTS OF THE GHRELIN RECEPTOR Pfizer Inc. (US) 2013-01-23 EP claimed
WO-2011114271-A1 2,3 DIHYDRO-1H-INDEN-1-YL- 2,7-DIAZASPIRO [3.6] NONANE DERIVATIVES AND THEIR USE AS ANTAGONISTS OR INVERSE AGONISTS OF THE GHRELIN RECEPTOR PFIZER INC. (US) 2011-09-22 WO claimed