SCHEMBL25248482

SCHEMBL25248482

O=[N+]([O-])c1cccc2c1oc1ccc(Br)cc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 5/20 0.55
GABRD O14764 5/20 0.55
GABRA1 P14867 5/20 0.55
GABRB1 P18505 5/20 0.55
GABRG2 P18507 5/20 0.55
GABRB3 P28472 5/20 0.55
GABRA5 P31644 5/20 0.55
GABRA3 P34903 5/20 0.55
GABRA2 P47869 5/20 0.55
GABRB2 P47870 5/20 0.55
GABRA4 P48169 5/20 0.55
GABRE P78334 5/20 0.55
GABRA6 Q16445 5/20 0.55
GABRG1 Q8N1C3 5/20 0.55
GABRG3 Q99928 5/20 0.55
GABRQ Q9UN88 5/20 0.55
GPR35 Q9HC97 1/20 0.47
MEN1 O00255 2/20 0.47
MAPT P10636 2/20 0.47
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17917509 0.81 KMT2A (0.54) GPR35MEN1MAPTKMT2AGAA
SCHEMBL8816924 0.77 GABRA1 (0.53) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL15497548 0.77 GABRP (0.50) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL23436651 0.77 GABRA1 (0.53) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL12396554 0.76 GABRP (0.44) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2370924 0.75 GABRP (0.46) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL3385902 0.74 MAOA (0.57) GPR35MEN1MAPTKMT2AGAA
SCHEMBL18862541 0.73 GPR35 (0.47) GPR35MEN1MAPTKMT2AGAA
SCHEMBL25290758 0.73 MAPT (0.42) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL19346715 0.73 TP53 (0.44) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023121238-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVE COMPOUND AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME (주)메디픽 2023-06-29 WO disclosed