SCHEMBL25344128

SCHEMBL25344128

CC(C)(C)OC(=O)NCCCn1cnc2ccc(F)c(Br)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.41
DYRK1A Q13627 1/20 0.40
BRD4 O60885 2/20 0.39
STK17B O94768 1/20 0.39
STK17A Q9UEE5 1/20 0.39
CA12 O43570 4/20 0.38
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA9 Q16790 4/20 0.38
PDPK1 O15530 1/20 0.38
CCNB2 O95067 1/20 0.38
PRKCB P05771 1/20 0.38
CDK1 P06493 1/20 0.38
LYN P07948 1/20 0.38
CCNB1 P14635 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
GSK3B P49841 1/20 0.38
RPS6KA3 P51812 1/20 0.38
CCNA1 P78396 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30568519 1.00 DRD2 (0.41) DRD2DYRK1ABRD4STK17BSTK17A
SCHEMBL25343224 0.83 PRPS1 (0.43) DRD2DYRK1ABRD4STK17BSTK17A
SCHEMBL25344478 0.81 DYRK1A (0.40) DRD2DYRK1ABRD4STK17BSTK17A
SCHEMBL25344380 0.80 SSTR4 (0.35) PDPK1CPB2
SCHEMBL30568621 0.80 SSTR4 (0.35) PDPK1CPB2
SCHEMBL31439941 0.80 MAOA (0.42) DRD2BRD4CA12CA1CA2
SCHEMBL25341649 0.79 DRD2 (0.46) DRD2BRD4CA12CA1CA2
SCHEMBL30568582 0.79 DYRK1A (0.47) DRD2DYRK1ABRD4STK17BSTK17A
SCHEMBL25342761 0.79 DYRK1A (0.47) DRD2DYRK1ABRD4STK17BSTK17A
SCHEMBL31440035 0.79 CAMK2D (0.46) DRD2DYRK1ABRD4STK17BSTK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023148129-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2023-08-10 WO disclosed