Isofezolac

Isofezolac

SCHEMBL25481

O=C(O)Cc1c(-c2ccccc2)c(-c2ccccc2)nn1-c1ccccc1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 3/20 0.52
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
FABP3 P05413 3/20 0.47
FABP4 P15090 3/20 0.47
FABP5 Q01469 2/20 0.45
FABP1 P07148 1/20 0.45
PTGIR P43119 1/20 0.44
DRD2 P14416 1/20 0.44
POLB P06746 2/20 0.43
PTGES O14684 1/20 0.42
ALOX5 P09917 1/20 0.42
RPA1 P27694 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SRC P12931 1/20 0.42
BRAF P15056 1/20 0.42
KDR P35968 1/20 0.42
LMNA P02545 1/20 0.42
PTGS2 P35354 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13013589 0.88 POLB (0.58) ALDH1A1KDM4EMEN1KMT2AFABP3
SCHEMBL3478412 0.88 MEN1 (0.48) ALDH1A1KDM4EMEN1KMT2AFABP3
SCHEMBL8766292 0.79 NPC1 (0.45) MEN1KMT2AFABP3FABP4SMN1; SMN2
SCHEMBL20054832 0.79 FABP4 (0.53) ALDH1A1KDM4EMEN1KMT2AFABP3
Bufezolac SCHEMBL287215 0.79 PTGIR (0.45) ALDH1A1KDM4EFABP3FABP4FABP5
SCHEMBL28345333 0.78 NPC1 (0.53) ALDH1A1KDM4EMEN1KMT2ADRD2
Isofezolac SCHEMBL2984804 0.78 CHRM1 (0.53) ALDH1A1ALOX5LMNAPTGS2PTGS1
SCHEMBL15489423 0.77 THRB (0.42) ALDH1A1KDM4EMEN1KMT2AFABP3
Trifezolac SCHEMBL11182574 0.77 KDM4E (0.51) ALDH1A1KDM4EMEN1KMT2APTGIR
SCHEMBL11724848 0.76 ALDH1A1 (0.50) ALDH1A1KDM4EMEN1KMT2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3097 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4470565-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT OnQuality Pharmaceuticals China Ltd. (CN) 2024-12-04 EP claimed
CN-118742325-A Methods for preventing or treating diseases or conditions associated with antineoplastic agents 上海岸阔医药科技有限公司 2024-10-01 CN claimed
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
WO-2023142996-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT 上海岸阔医药科技有限公司 2023-08-03 WO claimed
EP-4034087-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS Research Inc. (CA) 2022-08-03 EP claimed
US-20220218611-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS RESEARCH INC. (CA) 2022-07-14 US claimed
EP-3998932-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS Parsons, C. Lowell (US) 2022-05-25 EP claimed
US-20210145763-A1 LOW THC HEMP EXTRACT AND METHOD OF TREATMENT OR PREVENTION OF AN EYE DISEASE EYE CO PTY LTD. (AU) 2021-05-20 US claimed
WO-2021056106-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS RESEARCH INC. (CA) 2021-04-01 WO claimed
EP-3773651-A1 LOW THC HEMP EXTRACT AND METHOD OF TREATMENT OR PREVENTION OF AN EYE DISEASE Eye Co Pty Ltd. (AU) 2021-02-17 EP claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
US-5643943-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS FOR VASCULAR INFLAMMATION ALCON LABORATORIES, INC. (US) 1997-07-01 US claimed
WO-1997010236-A1 ESTERS OF NON-STEROIDAL ANTI-INFLAMMATORY CARBOXYLIC ACIDS ALCON LABORATORIES, INC. (US) 1997-03-20 WO claimed
EP-0759750-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO, Howard, K. (US) 1997-03-05 EP claimed
US-5607966-A BENZOFURAN OR BENZOPYRAN DERIVATIVES ALCON LABORATORIES, INC. (US) 1997-03-04 US claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
WO-1996020187-A2 ESTERS AND AMIDES OF NON-STEROIDAL ANTI-INFLAMMATORY CARBOXYLIC ACIDS WHICH MAY BE USED AS ANTI-OXIDANTS, 5-LIPOXYGENASE INHIBITORS AND NON-STEROIDAL ANTI-INFLAMMATORY PRODUCTS ALCON LABORATORIES, INC. (US) 1996-07-04 WO claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1995031194-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1995-11-23 WO claimed