Bufezolac

Bufezolac

SCHEMBL287215

CC(C)Cn1nc(-c2ccccc2)c(-c2ccccc2)c1CC(=O)O

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 1/20 0.45
PTGDR2 Q9Y5Y4 6/20 0.43
FABP4 P15090 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HSD17B10 Q99714 1/20 0.42
ALOX15 P16050 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
FABP3 P05413 3/20 0.41
TP53 P04637 1/20 0.41
FABP5 Q01469 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23402853 0.79 SMN1; SMN2 (0.41) PTGIRFABP4SMN1; SMN2HSD17B10ALOX15
Isofezolac SCHEMBL25481 0.79 ALDH1A1 (0.52) PTGIRPTGDR2FABP4SMN1; SMN2KDM4E
SCHEMBL6608161 0.76 SMN1; SMN2 (0.42) PTGIRFABP4SMN1; SMN2HSD17B10ALOX15
SCHEMBL23403471 0.74 FYN (0.40) SMN1; SMN2HSD17B10ALOX15KDM4EALDH1A1
SCHEMBL23400022 0.73 CASP1 (0.40) FABP4HSD17B10ALOX15KDM4EALDH1A1
SCHEMBL23399567 0.73 RAB9A (0.43) PTGIRSMN1; SMN2
SCHEMBL23403196 0.73 RAB9A (0.43) PTGIRSMN1; SMN2
SCHEMBL8890041 0.71 CSF1R (0.46) PTGIRSMN1; SMN2HSD17B10ALOX15KDM4E
SCHEMBL23400212 0.71 CYP1A2 (0.41) SMN1; SMN2HSD17B10ALOX15KDM4EALDH1A1
SCHEMBL23399087 0.71 MEN1 (0.40) KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 673 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20120183600-A1 NOVEL COMPOSITION FOR TREATING METABOLIC SYNDROME AND OTHER CONDITIONS CHEN CHIEN-HUNG (US) 2012-07-19 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
US-20080234380-A1 Compositions and method for treatment of chronic inflammatory diseases SHAPIRO HOWARD K 2008-09-25 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20050090553-A1 Compositions and method for treatment of chronic inflammatory diseases SECANT PHARMA, LLC 2005-04-28 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
EP-0759750-A4 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1998-05-27 EP claimed
EP-0759750-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO, Howard, K. (US) 1997-03-05 EP claimed
WO-1995031194-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1995-11-23 WO claimed
US-20250304667-A1 COMPLEMENT COMPONENT C5 ANTIBODIES ALLERGAN INC (US) 2025-10-02 US disclosed
EP-3693381-B1 LIGAND BINDING MOLECULES AND USES THEREOF VEGENICS PTY LTD (AU) 2025-09-03 EP disclosed
US-20250161402-A1 THERAPEUTIC COMPOSITIONS FOR THE TREATMENT OF DRY EYE DISEASE SCHEPENS EYE RES INST (US) 2025-05-22 US disclosed
EP-0123541-A1 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1984-10-31 EP disclosed
EP-0084822-A2 Diphosphonic acid derivatives and pharmaceutical preparations containing them SCHERING AKTIENGESELLSCHAFT (DE) 1983-08-03 EP disclosed
US-4391814-A Derivatives of antiphlogistically effective carboxylic acids, their preparation and medicinal use SCHERING AKTIENGESELLSCHAFT (DE) 1983-07-05 US disclosed
EP-0054812-A1 Derivatives of antiphlogistically active carboxylic acids, their preparation and medical application SCHERING AKTIENGESELLSCHAFT (DE) 1982-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050090553-A1 Compositions and method for treatment of chronic inflammatory diseases PCCA, HMGB1, PTGES PTGIR 439/4885PTGDR2 411/4885FABP4 157/4885
US-20080234380-A1 Compositions and method for treatment of chronic inflammatory diseases HMGB1, PCCA, QSOX1 PTGIR 441/4885PTGDR2 359/4885FABP4 202/4885
US-20250161402-A1 THERAPEUTIC COMPOSITIONS FOR THE TREATMENT OF DRY EYE DISEASE CRYAB, CRYAA, FUCA2 PTGIR 1161/4885PTGDR2 831/4885FABP4 644/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.