SCHEMBL254933

SCHEMBL254933

O=C1CCc2cccc3cccc1c23

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.68
KDM4E B2RXH2 4/20 0.68
HPGD P15428 3/20 0.68
HSD17B10 Q99714 4/20 0.56
LMNA P02545 2/20 0.56
TYMS P04818 6/20 0.56
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
PARP1 P09874 2/20 0.52
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
USP2 O75604 2/20 0.51
S100A4 P26447 1/20 0.51
CES1 P23141 2/20 0.46
CES2 O00748 1/20 0.46
BCHE P06276 1/20 0.46
MCL1 Q07820 1/20 0.46
CYP2A6 P11509 1/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30067536 1.00 ALDH1A1 (0.68) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL16230011 0.87 ALDH1A1 (0.61) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL975376 0.81 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL29383750 0.81 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDHSD17B10LMNA
Acenaphthene SCHEMBL3416108 0.77 TSHR (0.57) ALDH1A1KDM4EHPGDHSD17B10LMNA
Acenaphthene SCHEMBL9017 0.77 TSHR (0.57) ALDH1A1KDM4EHPGDHSD17B10LMNA
Acenaphthene SCHEMBL1162573 0.77 TSHR (0.57) ALDH1A1KDM4EHPGDHSD17B10LMNA
Acenaphthene SCHEMBL29386207 0.77 TSHR (0.57) ALDH1A1KDM4EHPGDHSD17B10LMNA
Acenaphthene SCHEMBL598252 0.77 TSHR (0.57) ALDH1A1KDM4EHPGDHSD17B10LMNA
Acenaphthene SCHEMBL28028969 0.77 TSHR (0.57) ALDH1A1KDM4EHPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 162 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014179528-A2 COMPOSITIONS AND METHODS TO IMPROVE THE THERAPEUTIC BENEFIT OF SUBOPTIMALLY ADMINISTERED CHEMICAL COMPOUNDS INCLUDING SUBSTITUTED NAPHTHALIMIDES SUCH AS AMONAFIDE FOR THE TREATMENT OF IMMUNOLOGICAL, METABOLIC, INFECTIOUS, AND BENIGN OR NEOPLASTIC HYPERPROLIFERATIVE DISEASE CONDITIONS BROWN DENNIS M (US) 2014-11-06 WO claimed
JP-3119718-A None JP disclosed
EP-4376822-A1 TREATING CANCERS WITH COMBINATIONS OF PARP INHIBITOR AND ACYLFULVENES Lantern Pharma Inc. (US) 2024-06-05 EP disclosed
US-20240156808-A1 Compositions and methods to improve the therapeutic benefit of suboptimally chemical compounds and biological therapies including substituted camptothecins such as irinotecan and topotecan for the treatment of benign and neoplastic hyperproliferative disease conditions, infections, inflammatory and immunological diseases EDISON ONCOLOGY (US) 2024-05-16 US disclosed
US-11913884-B2 Visible light-activated dyes and methods of use thereof WILLIAM MARSH RICE UNIVERSITY (US) 2024-02-27 US disclosed
EP-4297746-A2 COMPOSITIONS AND METHODS TO IMPROVE THE THERAPEUTIC BENEFIT OF SUBOPTIMALLY ADMINISTERED COMPOUNDS AND THERAPIES FOR THE TREATMENT OF DISEASES Edison Oncology (US) 2024-01-03 EP disclosed
US-11768434-B2 Polymer having a structure of polyamide, polyamide-imide, or polyimide, photosensitive resin composition, patterning process, photosensitive dry film, and protective film for electric and electronic parts SHIN-ETSU CHEMICAL CO., LTD. (JP) 2023-09-26 US disclosed
US-20230133044-A1 THERAPEUTIC BENEFIT OF SUBOPTIMALLY ADMINISTERED CHEMICAL COMPOUNDS BROWN DENNIS M (US) 2023-05-04 US disclosed
WO-2023069727-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF HYPERPROLIFERATIVE, INFLAMMATORY, AND IMMUNOLOGICAL DISEASES, AND INFECTIONS EDISON ONCOLOGY (US) 2023-04-27 WO disclosed
WO-2023010119-A1 TREATING CANCERS WITH COMBINATIONS OF PARP INHIBITOR AND ACYLFULVENES LANTERN PHARMA INC. (US) 2023-02-02 WO disclosed
EP-0281381-B1 ELECTROLUMINESCENT DEVICE WITH MODIFIED THIN FILM LUMINESCENT ZONE EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1992-07-15 EP disclosed
JP-H03119718-A FORMATION OF RESIST PATTERN OKI ELECTRIC IND CO LTD 1991-05-22 JP disclosed
US-4933948-A Inclusion compound of cyclodextrin and fluorescent dye EASTMAN KODAK COMPANY (US) 1990-06-12 US disclosed
US-4927927-A Fluorescent dyes and biological and analytical uses thereof EASTMAN KODAK COMPANY (US) 1990-05-22 US disclosed
EP-0349265-A2 Electroluminescent devices EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1990-01-03 EP disclosed
US-4812393-A ANALYTICAL DETERMINATION OF MICROORGANISMS EASTMAN KODAK COMPANY (US) 1989-03-14 US disclosed
EP-0281381-A2 Electroluminescent device with modified thin film luminescent zone EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1988-09-07 EP disclosed
US-4769292-A Electroluminescent device with modified thin film luminescent zone EASTMAN KODAK COMPANY (US) 1988-09-06 US disclosed
EP-0231127-A2 Composition, element and method using polymeric mordants to increase the intensity of rigid fluorescent dyes EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1987-08-05 EP disclosed
EP-0231126-A2 Fluorescent dyes and biological and analytical uses thereof EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1987-08-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133044-A1 THERAPEUTIC BENEFIT OF SUBOPTIMALLY ADMINISTERED CHEMICAL COMPOUNDS UNG, DPYD, TPMT ALDH1A1 379/4885KDM4E 714/4885HPGD 958/4885
US-11913884-B2 Visible light-activated dyes and methods of use thereof HCCS, CLTB, ALDH1A2 ALDH1A1 311/4885KDM4E 3264/4885HPGD 2058/4885
US-20240156808-A1 Compositions and methods to improve the therapeutic benefit of suboptimally chemical compounds and biological therapies including substituted camptothecins such as irinotecan and topotecan for the treatment of benign and neoplastic hyperproliferative disease conditions, infections, inflammatory and immunological diseases TOP2A, TOP2B, TOP1 ALDH1A1 3441/4885KDM4E 4039/4885HPGD 672/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.