SCHEMBL254955

SCHEMBL254955

Nc1ccc(-c2ccc(C(=O)Oc3c(F)c(F)c(F)c(F)c3F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
LMNA P02545 2/20 0.47
CYP1A2 P05177 2/20 0.47
MAOA P21397 2/20 0.47
SENP1 Q9P0U3 1/20 0.45
F2 P00734 2/20 0.43
PRSS1 P07477 2/20 0.43
PRSS2 P07478 2/20 0.43
PRSS3 P35030 2/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
TSHR P16473 2/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
PDE4D Q08499 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
PHLPP2 Q6ZVD8 1/20 0.41
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889497 0.85 SENP1 (0.47) SENP1KMT2ATSHRALDH1A1NPC1
SCHEMBL15235763 0.83 LMNA (0.41) CYP3A4LMNACYP1A2MAOAF2
SCHEMBL27682095 0.80 PARP10 (0.53) CYP3A4SENP1F2PRSS1PRSS2
SCHEMBL23235066 0.80 RAB9A (0.49) CYP1A2SENP1PKMKMT2ANPC1
SCHEMBL10021501 0.78 PRSS1 (0.65) CYP3A4LMNACYP1A2MAOAF2
SCHEMBL22310501 0.78 PRSS1 (0.65) CYP3A4LMNACYP1A2MAOAF2
SCHEMBL8712521 0.78 CA1 (0.55) PRSS1KMT2ATSHRALDH1A1NPC1
SCHEMBL15712039 0.78 TDP1 (0.55) LMNACYP1A2PRSS1PKMKMT2A
SCHEMBL3143505 0.78 PRSS1 (0.65) CYP3A4LMNACYP1A2MAOAF2
SCHEMBL10126445 0.78 SENP1 (0.59) LMNACYP1A2SENP1PKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed