SCHEMBL25515560

SCHEMBL25515560

CON(C)C(=O)c1ccn2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 1/20 0.35
MLYCD O95822 1/20 0.34
ALDH1A1 P00352 7/20 0.34
CYP3A4 P08684 2/20 0.34
LPAR5 Q9H1C0 1/20 0.34
KDM4E B2RXH2 7/20 0.33
HPGD P15428 5/20 0.33
GAA P10253 4/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NR4A2 P43354 1/20 0.33
HTT P42858 2/20 0.32
POLB P06746 1/20 0.32
CLK1 P49759 1/20 0.32
DYRK1A Q13627 1/20 0.32
DYRK1B Q9Y463 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25515031 0.90 MLYCD (0.36) TRPM8MLYCDALDH1A1CYP3A4LPAR5
SCHEMBL28974225 0.83 KMT2A (0.43) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL26127613 0.79 CLK1 (0.45) ALDH1A1CYP3A4LPAR5KDM4EHPGD
SCHEMBL26128828 0.78 MLYCD (0.35) TRPM8MLYCDALDH1A1LPAR5KDM4E
SCHEMBL26128304 0.78 CLK1 (0.41) ALDH1A1LPAR5KDM4EHPGDGAA
SCHEMBL3983002 0.77 NR4A2 (0.50) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL26125608 0.76 LPAR5 (0.40) LPAR5GAAHTTPOLBCLK1
SCHEMBL9231407 0.74 BAZ2B (0.41) ALDH1A1KDM4EHPGDGAAPOLB
SCHEMBL27516303 0.74 FNTA (0.39) ALDH1A1CYP3A4KDM4EHPGDGAA
SCHEMBL18137568 0.74 QPCT (0.44) TRPM8MLYCDALDH1A1CYP3A4LPAR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250042900-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION TACTOGEN INC (US) 2025-02-06 US disclosed
EP-4499058-A2 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION Tactogen Inc. (US) 2025-02-05 EP disclosed
US-20240308999-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR MENTAL ENHANCEMENT TACTOGEN INC (US) 2024-09-19 US disclosed
EP-4426291-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR MENTAL ENHANCEMENT Tactogen Inc. (US) 2024-09-11 EP disclosed
WO-2023183613-A2 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION TACTOGEN INC (US) 2023-09-28 WO disclosed
WO-2023183613-A2 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION TACTOGEN INC (US) 2023-09-28 WO disclosed
WO-2023081306-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR MENTAL ENHANCEMENT TACTOGEN INC (US) 2023-05-11 WO disclosed
WO-2023081306-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR MENTAL ENHANCEMENT TACTOGEN INC (US) 2023-05-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240308999-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR MENTAL ENHANCEMENT PNMT, HTR5A, HTR4 TRPM8 506/4885MLYCD 1067/4885ALDH1A1 4486/4885
US-20250042900-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION TPH2, TPH1, IDO2 TRPM8 1083/4885MLYCD 638/4885ALDH1A1 2187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.