SCHEMBL255347

SCHEMBL255347

NC(=O)c1cc2cccnc2nc1Cc1ccc(C2CCOCC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SYK P43405 5/20 0.38
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
MAPK1 P28482 3/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
PARP1 P09874 2/20 0.34
CNR1 P21554 3/20 0.34
CNR2 P34972 3/20 0.34
GRM4 Q14833 1/20 0.33
KCNH2 Q12809 1/20 0.33
ATM Q13315 1/20 0.33
ATR Q13535 1/20 0.33
ROCK2 O75116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL253123 0.78 SYK (0.42) SYKIRAK4KCNH2ROCK2
SCHEMBL617662 0.75 HTT (0.46) MAPK1
SCHEMBL252708 0.74 MKNK1 (0.48) SYKPARP1
SCHEMBL253870 0.72 CYP11B1 (0.52) CYP11B1CYP11B2IRAK4PARP1
SCHEMBL255348 0.71 NAMPT (0.52) MAPK1
SCHEMBL252286 0.71 PARP1 (0.41) PARP1
SCHEMBL253705 0.70 AURKA (0.47) PARP1
SCHEMBL28566904 0.70 LMNA (0.45)
SCHEMBL253898 0.69 SYK (0.41) SYKIRAK4PARP1
SCHEMBL5083476 0.67 OPRL1 (0.46) CYP11B1CYP11B2MAPK1PARP1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP claimed