SCHEMBL252286

SCHEMBL252286

NC(=O)c1cc2cccnc2nc1Cc1ccc(-c2ccccc2C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
SCN9A Q15858 5/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
SLC6A7 Q99884 1/20 0.39
SLC13A5 Q86YT5 1/20 0.39
CD38 P28907 1/20 0.38
SUCNR1 Q9BXA5 4/20 0.38
FFAR4 Q5NUL3 1/20 0.38
GRM2 Q14416 1/20 0.38
RPS6KB1 P23443 1/20 0.38
CAMKK2 Q96RR4 1/20 0.37
CDC7 O00311 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
DBF4 Q9UBU7 1/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
DHODH Q02127 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL253705 0.78 AURKA (0.47) PARP1RPS6KB1
SCHEMBL252708 0.78 MKNK1 (0.48) PARP1DHODH
SCHEMBL617276 0.76 HTT (0.50) SCN9ASUCNR1PPARA
SCHEMBL253870 0.75 CYP11B1 (0.52) PARP1
SCHEMBL253233 0.75 SYK (0.40) RPS6KB1PPARGPPARA
SCHEMBL248207 0.75 CSF1R (0.43) RPS6KB1CDK2
SCHEMBL253123 0.73 SYK (0.42)
SCHEMBL28566904 0.72 LMNA (0.45)
SCHEMBL252287 0.71 STAMBP (0.51) SCN9ASUCNR1
SCHEMBL253898 0.71 SYK (0.41) PARP1SUCNR1CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP claimed
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP disclosed