SCHEMBL25577924

SCHEMBL25577924

COc1ccc(CN(Cc2ccc(OC)cc2)S(=O)(=O)c2ccc(CBr)cc2F)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
APLNR P35414 3/20 0.52
TAS2R14 Q9NYV8 12/20 0.52
L3MBTL1 Q9Y468 1/20 0.50
KCNA5 P22460 1/20 0.47
PTGES O14684 1/20 0.45
TAS2R8 Q9NYW2 1/20 0.45
CXCR3 P49682 1/20 0.45
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31149207 0.88 L3MBTL1 (0.52) APLNRTAS2R14L3MBTL1KCNA5
SCHEMBL31149228 0.88 APLNR (0.51) APLNRTAS2R14L3MBTL1KCNA5PTGES
SCHEMBL4183685 0.88 L3MBTL1 (0.52) APLNRTAS2R14L3MBTL1KCNA5
SCHEMBL31149689 0.88 APLNR (0.51) APLNRTAS2R14L3MBTL1KCNA5PTGES
SCHEMBL31149661 0.88 TAS2R14 (0.54) APLNRTAS2R14L3MBTL1KCNA5PTGES
SCHEMBL25578370 0.87 TAS2R14 (0.55) APLNRTAS2R14PTGESTAS2R8CXCR3
SCHEMBL25578283 0.84 APLNR (0.52) APLNRTAS2R14L3MBTL1PTGESTAS2R8
SCHEMBL30219708 0.84 APLNR (0.52) APLNRTAS2R14L3MBTL1PTGESTAS2R8
SCHEMBL31149206 0.83 TAS2R14 (0.57) APLNRTAS2R14PTGESTAS2R8CXCR3
SCHEMBL31149813 0.83 TAS2R14 (0.66) TAS2R14PTGESTAS2R8CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4695242-A1 NOVEL SUBSTITUTED PYRROLE COMPOUNDS, COMPOSITIONS COMPRISING THE SUBSTITUTED PYRROLE COMPOUND, AND METHODS OF USE THEREOF Meta Pharmaceuticals (HK) Limited (HK) 2026-02-18 EP disclosed
CN-115996924-B Substituted pyrazolyl compounds and methods of use thereof 诺华医药股份公司 2025-03-07 CN disclosed
WO-2024212907-A1 NOVEL SUBSTITUTED PYRROLE COMPOUNDS, COMPOSITIONS COMPRISING THE SUBSTITUTED PYRROLE COMPOUND, AND METHODS OF USE THEREOF META PHARMACEUTICALS (HK) LIMITED (CN) 2024-10-17 WO disclosed
WO-2024212024-A1 NOVEL SUBSTITUTED PYRROLE COMPOUNDS, COMPOSITIONS COMPRISING THE SUBSTITUTED PYRROLE COMPOUND, AND METHODS OF USE THEREOF META PHARMACEUTICALS (HK) LIMITED (CN) 2024-10-17 WO disclosed
US-20230183228-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS AND METHODS OF USE THEREOF NOVARTIS PHARMA AG (CH) 2023-06-15 US disclosed
CN-115996924-A Substituted pyrazolyl compounds and methods of use thereof 奇努克医疗加拿大公司 2023-04-21 CN disclosed
EP-4153586-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS AND METHODS OF USE THEREOF Chinook Therapeutics Canada, Inc. (CA) 2023-03-29 EP disclosed
EP-4153585-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS AND METHODS OF USE THEREOF Chinook Therapeutics Canada, Inc. (CA) 2023-03-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230183228-A1 SUBSTITUTED PYRAZOLYL COMPOUNDS AND METHODS OF USE THEREOF LDHA, LDHB, XDH APLNR 4775/4885TAS2R14 3827/4885L3MBTL1 1002/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.