SCHEMBL25599642

SCHEMBL25599642

COCc1cc2c(cc1[N+](=O)[O-])nc(N1CCCC(F)C1)n2C

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.37
HSD11B1 P28845 1/20 0.35
DPP4 P27487 1/20 0.34
ALDH1A1 P00352 3/20 0.33
PKM P14618 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 1/20 0.33
CYP2D6 P10635 1/20 0.33
GAA P10253 1/20 0.32
OPRM1 P35372 1/20 0.32
MAPT P10636 2/20 0.32
CHRM3 P20309 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25599264 0.84 KCNH2 (0.44) KCNH2HSD11B1ALDH1A1PKMMEN1
SCHEMBL25599685 0.83 KCNH2 (0.37) KCNH2HSD11B1ALDH1A1PKMMEN1
SCHEMBL25599242 0.83 ALDH1A1 (0.40) KCNH2HSD11B1ALDH1A1PKMMEN1
SCHEMBL25681759 0.83 DPP4 (0.36) KCNH2DPP4CHRM3PDE4APDE4B
SCHEMBL25599724 0.83 MAPT (0.45) ALDH1A1PKMMEN1KMT2ALMNA
SCHEMBL25599801 0.80 MAPT (0.42) KCNH2DPP4ALDH1A1MEN1KMT2A
SCHEMBL25599269 0.79 ALDH1A1 (0.35) KCNH2HSD11B1ALDH1A1PKMMEN1
SCHEMBL25599637 0.76 UCHL3 (0.38) DPP4
SCHEMBL25216705 0.75 MET (0.33) CYP2D6MAPT
SCHEMBL30464393 0.75 MET (0.33) CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023102184-A1 BICYCLIC AMINE COMPOUNDS AS CDK12 INHIBITORS INCYTE CORPORATION (US) 2023-06-08 WO disclosed