SCHEMBL25663232

SCHEMBL25663232

COC(=O)c1c(OC)c(=O)c(C(N)=O)cn1CC=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.34
PDE3B Q13370 3/20 0.33
PDE3A Q14432 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
BRD4 O60885 1/20 0.33
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
KDM4E B2RXH2 3/20 0.31
POLB P06746 1/20 0.31
ALDH1A1 P00352 3/20 0.31
HPGD P15428 2/20 0.31
MAPK10 P53779 1/20 0.31
KMT2A Q03164 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239239 0.88 RAB9A (0.41) NR4A2SMN1; SMN2LMNAMAPTBRD4
SCHEMBL18896381 0.83 PDE3B (0.36) NR4A2PDE3BPDE3ASMN1; SMN2LMNA
SCHEMBL17967309 0.82 PDE3B (0.33) NR4A2PDE3BPDE3ASMN1; SMN2LMNA
SCHEMBL18010785 0.79 ALDH1A1 (0.47) NR4A2SMN1; SMN2LMNAMAPTBRD4
SCHEMBL15084306 0.79 KDM4E (0.43) LMNAMAPTRAB9AKDM4EALDH1A1
SCHEMBL17967300 0.77 KMT2A (0.41) NR4A2LMNARAB9ANPC1KDM4E
SCHEMBL2601037 0.77 PLA2G4A (0.38) NR4A2SMN1; SMN2LMNAMAPTBRD4
SCHEMBL17928514 0.75 TSHR (0.39) NR4A2LMNABRD4RAB9AKDM4E
SCHEMBL16453350 0.74 PDE10A (0.53)
SCHEMBL19041053 0.74 LMNA (0.45) NR4A2SMN1; SMN2LMNAMAPTBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023083162-A1 POLYCYCLIC CARBAMOYL PYRIDONE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION THEREOF 南京艾迪医药科技有限公司 2023-05-19 WO disclosed