SCHEMBL2567237

SCHEMBL2567237

CCOC(=O)Oc1nc(N)cn1CC1CC1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
JAK1 P23458 9/20 0.38
JAK2 O60674 5/20 0.38
TYK2 P29597 5/20 0.38
OPRD1 P41143 1/20 0.36
JAK3 P52333 2/20 0.36
SRC P12931 1/20 0.33
KCNH2 Q12809 1/20 0.33
DYRK1A Q13627 3/20 0.33
GRK6 P43250 1/20 0.33
PTGER4 P35408 1/20 0.33
ICMT O60725 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2570796 0.82 MITF (0.49) JAK1JAK2TYK2OPRD1JAK3
SCHEMBL1594682 0.80 LMNA (0.45) LMNAJAK1JAK2TYK2OPRD1
SCHEMBL2570702 0.76 ADORA3 (0.39) LMNA
Hydrochloric Acid SCHEMBL23389304 0.72 CYP11B2 (0.35) LMNAKCNH2DYRK1AICMT
SCHEMBL14786484 0.72 CYP11B2 (0.35) LMNAKCNH2DYRK1AICMT
SCHEMBL14786459 0.71 POLB (0.46) LMNA
SCHEMBL7607398 0.68 LMNA (0.43) LMNAPTGER4ICMT
Hydrochloric Acid SCHEMBL23389330 0.66 MEN1 (0.35) LMNAJAK2KCNH2DYRK1A
SCHEMBL23389350 0.66 MAPT (0.38) LMNAOPRD1DYRK1A
SCHEMBL23389316 0.66 MEN1 (0.35) LMNAJAK2KCNH2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2755964-B1 SULFONIC ACID SALTS OF HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLES AICURIS ANTI INFECTIVE CURES GMBH (DE) 2016-06-22 EP disclosed
EP-2755964-A1 SULFONIC ACID SALTS OF HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLES AiCuris GmbH & Co. KG (DE) 2014-07-23 EP disclosed
WO-2013037812-A1 SULFONIC ACID SALTS OF HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLES AICURIS GMBH & CO. KG (DE) 2013-03-21 WO disclosed
EP-1732901-B1 ANTIVIRAL 4-AMINOCARBONYLAMINO-SUBSTITUTED IMIDAZOLE COMPOUND AICURIS GMBH & CO KG (DE) 2011-11-02 EP disclosed
EP-1853582-B1 HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLES AICURIS GMBH & CO KG (DE) 2009-10-21 EP disclosed
EP-1853582-A2 HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLES AiCuris GmbH & Co. KG (DE) 2007-11-14 EP disclosed
EP-1732901-A1 ANTIVIRAL 4-AMINOCARBONYLAMINO-SUBSTITUTED IMIDAZOLE COMPOUND Bayer HealthCare AG (DE) 2006-12-20 EP disclosed
WO-2006089664-A2 HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLES AICURIS GMBH & CO. KG (DE) 2006-08-31 WO disclosed
WO-2005092865-A1 ANTIVIRAL 4-AMINOCARBONYLAMINO-SUBSTITUTED IMIDAZOLE COMPOUND BAYER HEALTHCARE AG (DE) 2005-10-06 WO disclosed