SCHEMBL25709673

SCHEMBL25709673

CCc1ccc(C(=N)C(C)CC)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
IDO1 P14902 2/20 0.41
PLK1 P53350 1/20 0.41
CHRM2 P08172 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
CHRM3 P20309 1/20 0.41
DRD3 P35462 1/20 0.41
OPRD1 P41143 1/20 0.41
KCNH2 Q12809 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
PLAU P00749 2/20 0.38
F2 P00734 1/20 0.38
PLG P00747 1/20 0.38
PLAT P00750 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19007619 0.79 LMNA (0.40) ALDH1A1SMN1; SMN2ADRA2BKCNH2F2
SCHEMBL23965631 0.78 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2IDO1PLK1TAS1R3
SCHEMBL6485939 0.73 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2IDO1PLK1TAS1R3
SCHEMBL26216411 0.73 PRSS1 (0.55) ALDH1A1SMN1; SMN2TAS1R3TAS1R1PRSS1
SCHEMBL10308978 0.72 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2IDO1PLK1TAS1R3
SCHEMBL13944771 0.70 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2IDO1PLK1TAS1R3
SCHEMBL1696572 0.70 PRSS1 (0.64) ALDH1A1SMN1; SMN2IDO1PLAUF2
SCHEMBL22901598 0.69 TAS1R3 (0.44) ALDH1A1SMN1; SMN2IDO1PLK1CHRM2
Hydrochloric Acid SCHEMBL11567719 0.68 PRSS1 (0.61) ALDH1A1SMN1; SMN2IDO1PLAUF2
SCHEMBL3129690 0.67 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2PLK1CHRM2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023114822-A1 BENZOTHIAZOLE, BENZOISOXAZOLE AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-06-22 WO disclosed