SCHEMBL3129690

SCHEMBL3129690

CCc1ccc(C(=O)C(C)C)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
CHRM2 P08172 1/20 0.54
CYP2D6 P10635 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
CHRM3 P20309 1/20 0.54
DRD3 P35462 1/20 0.54
OPRD1 P41143 1/20 0.54
KCNH2 Q12809 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
HRH3 Q9Y5N1 1/20 0.54
PLK1 P53350 1/20 0.53
TAS1R3 Q7RTX0 1/20 0.53
TAS1R1 Q7RTX1 1/20 0.53
KDM4E B2RXH2 1/20 0.48
DBH P09172 1/20 0.48
GAA P10253 1/20 0.48
RECQL P46063 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480603 0.84 KMT2A (0.58) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C
SCHEMBL3685675 0.84 KDM4E (0.50) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C
SCHEMBL9559796 0.83 ALDH1A1 (0.55) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C
SCHEMBL10730260 0.83 ALDH1A1 (0.55) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C
SCHEMBL16868406 0.83 ALDH1A1 (0.55) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C
SCHEMBL19520440 0.83 ALDH1A1 (0.55) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C
SCHEMBL9666038 0.83 PLK1 (0.56) ALDH1A1PLK1TAS1R3TAS1R1KDM4E
SCHEMBL10121174 0.83 KDM4E (0.62) ALDH1A1ADRA2BKCNH2KDM4EDBH
SCHEMBL12158530 0.83 SLC6A2 (0.49) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C
SCHEMBL9617195 0.82 CHRM2 (0.58) ALDH1A1CHRM2CYP2D6ADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000285-B1 7-ACYLAMINO-3-((3-(CARBOXYMETHYL) THIO-1 H-1,2,4-TRIAZOL-5-YL) THIOMETHYL)-3-CEPHEM-4-CARBOXYLIC ACID DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM SMITHKLINE BECKMAN CORPORATION (US) 1982-02-17 EP claimed
US-11872206-B2 Purified forms of rofecoxib, methods of manufacture and use Tremeau Pharmaceuticals, Inc. (US) 2024-01-16 US disclosed
US-11872206-B2 Purified forms of rofecoxib, methods of manufacture and use Tremeau Pharmaceuticals, Inc. (US) 2024-01-16 US disclosed
US-20230159569-A1 DUAL HDAC6/PROTEASOME INHIBITORS, AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-05-25 US disclosed
US-11576890-B2 Purified forms of rofecoxib, methods of manufacture and use Tremeau Pharmaceuticals, Inc. (US) 2023-02-14 US disclosed
US-11572364-B2 Pteridinone compounds and uses thereof VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-02-07 US disclosed
US-20210236455-A1 PURIFIED FORMS OF ROFECOXIB, METHODS OF MANUFACTURE AND USE Tremeau Pharmaceuticals, Inc. (US) 2021-08-05 US disclosed
EP-3789426-A1 POLYARYLETHER KETONE IMIDE SULFONE ADHESIVES The Boeing Company (US) 2021-03-10 EP disclosed
US-20180148453-A1 DIHYDROPYRAZOLOPYRIMIDINONE COMPOUNDS AS PDE2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-05-31 US disclosed
US-20170290928-A1 USE OF CHARGE-BALANCED IMAGING AGENTS FOR DETERMINING RENAL FUNCTION BETH ISRAEL DEACONESS MEDICAL CT INC (US) 2017-10-12 US disclosed
EP-0414207-B1 Method for preparing alpha-(-4-isobutylphenyl) propionic acid or its precursor NIPPON PETROCHEMICALS CO LTD (JP) 1994-08-03 EP disclosed
EP-0373362-B1 METHOD FOR PREPARING P-ISOBUTYLSTYRENE NIPPON PETROCHEMICALS COMPANY, LIMITED (JP) 1993-02-03 EP disclosed
US-5166419-A Multistage reaction by catalytic dehydrogenation and reaction with carbon monoxide NIPPON PETROCHEMICALS CO., LTD. (JP) 1992-11-24 US disclosed
EP-0273647-B1 COUMARAN DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-03-11 EP disclosed
EP-0423524-A2 Propiophenone derivatives and their preparation and pharmaceutical use MARUHO Co., Ltd. (JP) 1991-04-24 EP disclosed
EP-0414207-A2 Method for preparing alpha-(-4-isobutylphenyl) propionic acid or its precursor NIPPON PETROCHEMICALS CO., LTD. (JP) 1991-02-27 EP disclosed
EP-0373362-A1 Method for preparing p-isobutylstyrene NIPPON PETROCHEMICALS COMPANY, LIMITED (JP) 1990-06-20 EP disclosed
US-4857516-A Coumaran derivatives and their pharmaceutical use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-08-15 US disclosed
EP-0273647-A1 Coumaran derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-07-06 EP disclosed
US-4352748-A Novel acyl-polyalkylindan compounds and the use thereof as a base for perfume, as well as perfume compositions NAARDEN INTERNATIONAL N.V. (NL) 1982-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210236455-A1 PURIFIED FORMS OF ROFECOXIB, METHODS OF MANUFACTURE AND USE ITGA2B, F13B, F11 ALDH1A1 2666/4885CHRM2 1668/4885CYP2D6 576/4885
US-11872206-B2 Purified forms of rofecoxib, methods of manufacture and use ITGA2B, F13B, F11 ALDH1A1 2666/4885CHRM2 1668/4885CYP2D6 576/4885
US-11572364-B2 Pteridinone compounds and uses thereof DPYD, PKD1, TYMP ALDH1A1 569/4885CHRM2 4314/4885CYP2D6 1271/4885
US-20230159569-A1 DUAL HDAC6/PROTEASOME INHIBITORS, AND METHODS OF USE THEREOF HDAC6, PSMG3, PSMB2 ALDH1A1 2269/4885CHRM2 4843/4885CYP2D6 4748/4885
US-11576890-B2 Purified forms of rofecoxib, methods of manufacture and use ITGA2B, F13B, F11 ALDH1A1 2666/4885CHRM2 1668/4885CYP2D6 576/4885
US-20180148453-A1 DIHYDROPYRAZOLOPYRIMIDINONE COMPOUNDS AS PDE2 INHIBITORS PDE12, PDE2A, PDE4D ALDH1A1 635/4885CHRM2 543/4885CYP2D6 584/4885
US-20170290928-A1 USE OF CHARGE-BALANCED IMAGING AGENTS FOR DETERMINING RENAL FUNCTION ATP6V1B1, SLC8B1, PHOSPHO1 ALDH1A1 4754/4885CHRM2 2723/4885CYP2D6 4794/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.