SCHEMBL257205

SCHEMBL257205

COc1ccc(CN(Cc2ccc(OC)cc2)c2nc(-c3cccc(Br)c3)c(C(=O)c3ccccc3)s2)cc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.57
ADORA2A P29274 3/20 0.48
ADORA1 P30542 5/20 0.48
ADORA3 P0DMS8 4/20 0.48
HTT P42858 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
ALDH1A1 P00352 1/20 0.45
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
ACHE P22303 1/20 0.44
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTGDR2 Q9Y5Y4 3/20 0.42
KARS1 Q15046 1/20 0.42
RORB Q92753 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20286599 0.91 ALOX5 (0.67) ALOX5ADORA2AADORA1ADORA3HTT
SCHEMBL168009 0.89 ALOX5 (0.55) ALOX5ADORA2AADORA1ADORA3HTT
SCHEMBL4746033 0.87 ALOX5 (0.62) ALOX5ADORA2AADORA1ADORA3HTT
SCHEMBL4746826 0.80 ALOX5 (0.57) ALOX5ADORA2AADORA1ADORA3HTT
SCHEMBL168675 0.79 RORB (0.46) ALOX5LMNAMAPTPTGDR2RORB
SCHEMBL8154046 0.78 ALOX5 (0.52) ALOX5ADORA2AADORA1ADORA3HTT
SCHEMBL4746026 0.73 ADORA2A (0.49) ALOX5ADORA2AADORA1ADORA3HTT
SCHEMBL169403 0.66 RORC (0.58) ADORA2AADORA1ADORA3HTTNPSR1
SCHEMBL20969597 0.66 KARS1 (0.65) HTTPPARGPPARALMNAMAPT
SCHEMBL20969558 0.66 KARS1 (0.65) ALDH1A1PPARGPPARAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed