SCHEMBL257433

SCHEMBL257433

COc1ccccc1C(=O)c1sc(N)nc1-c1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RORB Q92753 14/20 0.72
RORC P51449 3/20 0.66
POLB P06746 1/20 0.57
ALDH1A1 P00352 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CDK5 Q00535 2/20 0.50
CDK5R1 Q15078 2/20 0.50
CFTR P13569 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL257260 0.83 RORB (0.60) RORBRORCPOLBALDH1A1HSD17B10
SCHEMBL1256222 0.82 RORB (0.60) RORBRORCPOLBALDH1A1HSD17B10
SCHEMBL27653923 0.82 ALDH1A1 (0.64) RORBRORCPOLBALDH1A1HSD17B10
SCHEMBL257269 0.80 RORB (0.60) RORBRORCALDH1A1HSD17B10
SCHEMBL257608 0.80 RORB (0.83) RORBRORCPOLBALDH1A1HSD17B10
SCHEMBL257375 0.80 RORB (0.60) RORBRORCPOLBALDH1A1HSD17B10
SCHEMBL19669120 0.78 ALDH1A1 (0.72) RORCPOLBALDH1A1HSD17B10
SCHEMBL4880192 0.78 FBP1 (0.67) RORB
SCHEMBL165773 0.78 ADORA3 (0.61) RORBPOLBALDH1A1HSD17B10
SCHEMBL256651 0.77 RORB (0.79) RORBRORCALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed