SCHEMBL257269

SCHEMBL257269

Nc1nc(-c2ccccc2)c(C(=O)c2ccccc2F)s1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORB Q92753 15/20 0.60
RORC P51449 1/20 0.54
ALDH1A1 P00352 3/20 0.53
HSD17B10 Q99714 1/20 0.53
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
MAPT P10636 1/20 0.50
CYP2C19 P33261 1/20 0.50
ADORA3 P0DMS8 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA1 P30542 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL256653 0.90 RORB (0.59) RORBRORCALDH1A1SMN1; SMN2MAPT
SCHEMBL257434 0.86 RORB (0.79) RORBRORC
SCHEMBL27653923 0.85 ALDH1A1 (0.64) RORBRORCALDH1A1HSD17B10SMN1; SMN2
SCHEMBL257375 0.83 RORB (0.60) RORBRORCALDH1A1HSD17B10CYP1A2
SCHEMBL257608 0.83 RORB (0.83) RORBRORCALDH1A1HSD17B10CYP1A2
SCHEMBL257260 0.83 RORB (0.60) RORBRORCALDH1A1HSD17B10CYP1A2
SCHEMBL256651 0.83 RORB (0.79) RORBRORCALDH1A1HSD17B10CYP1A2
SCHEMBL165773 0.81 ADORA3 (0.61) RORBALDH1A1HSD17B10SMN1; SMN2CYP1A2
SCHEMBL1255464 0.81 MEN1 (0.50) RORBRORCALDH1A1HSD17B10NPC1
SCHEMBL257433 0.80 RORB (0.72) RORBRORCALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed