SCHEMBL25751659

SCHEMBL25751659

COC(=O)c1[nH]c2ccc(Cl)cc2c1N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.58
ALDH1A1 P00352 6/20 0.58
HPGD P15428 5/20 0.58
GAA P10253 3/20 0.58
MAPT P10636 3/20 0.58
HSD17B10 Q99714 3/20 0.58
NPSR1 Q6W5P4 2/20 0.58
USP2 O75604 1/20 0.58
ALOX15 P16050 1/20 0.58
TUBB4A P04350 5/20 0.57
TUBB P07437 5/20 0.57
TUBA3C P0DPH7 5/20 0.57
TUBA1B P68363 5/20 0.57
TUBA4A P68366 5/20 0.57
TUBB4B P68371 5/20 0.57
TUBB3 Q13509 5/20 0.57
TUBB2A Q13885 5/20 0.57
TUBB8 Q3ZCM7 5/20 0.57
TUBA3E Q6PEY2 5/20 0.57
TUBA1A Q71U36 5/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538872 0.88 KDM4E (0.70) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL13758172 0.85 ALDH1A1 (0.76) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL23873802 0.84 ALDH1A1 (0.74) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL21465510 0.84 KDM4E (0.60) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL3253095 0.83 KDM4E (0.56) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL6308065 0.82 KDM4E (0.58) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL21465557 0.82 TUBB4A (0.65) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL31219205 0.81 MAP2 (0.66) KDM4EALDH1A1MAP2
SCHEMBL4332943 0.81 MAP2 (0.61) KDM4EALDH1A1MEN1KMT2AMAP2
SCHEMBL5402454 0.80 ALOX15 (0.60) KDM4EALDH1A1HPGDGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116390-A1 PYRIMIDINE-2(1H)-ONE-FUSED BICYCLIC COMPOUND HAVING MAT2A INHIBITORY ACTIVITY AND USE THEREOF 上海海和药物研究开发股份有限公司 2023-06-29 WO disclosed