SCHEMBL25759480

SCHEMBL25759480

Nc1ccc(F)c(S(=O)(=O)Nc2c(F)cc(Cl)cc2F)c1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CCR2 P41597 7/20 0.44
ALPL P05186 2/20 0.42
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ACLY P53396 2/20 0.40
PTK2B Q14289 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SGK1 O00141 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23846522 0.81 POLB (0.60) MEN1KMT2AALPLPOLBMAPT
SCHEMBL25754794 0.80 TSHR (0.50) MEN1KMT2ACCR2POLBPTK2B
SCHEMBL1805587 0.78 ALOX5AP (0.41) MEN1KMT2A
SCHEMBL25754828 0.77 SMN1; SMN2 (0.51) MEN1KMT2APOLBMAPTNPSR1
SCHEMBL23833706 0.77 NHERF1 (0.49) MEN1KMT2ACCR2MAPTTDP1
SCHEMBL25754792 0.76 SGK1 (0.52) MEN1KMT2APOLBMAPTNPSR1
SCHEMBL23847021 0.74 PKM (0.56) MEN1KMT2APOLBMAPTNPSR1
SCHEMBL22981720 0.74 MCL1 (0.48) MEN1KMT2AACLYSGK1
SCHEMBL29434895 0.74 MCL1 (0.48) MEN1KMT2AACLYSGK1
SCHEMBL3451784 0.72 L3MBTL1 (0.57) MEN1KMT2ACCR2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 MEN1 3902/4885KMT2A 4864/4885CCR2 3679/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.